[ASAP] Novel Serine-Arginine Protein Kinase Inhibitors for Treating Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00132 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 25, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Beyond 20 in the 21st Century: Prospects and Challenges of Non ‑canonical Amino Acids in Peptide Drug Discovery
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00037 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 24, 2023 Category: Chemistry Authors: Jennifer L. Hickey, Dan Sindhikara, Susan L. Zultanski, and Danielle M. Schultz Source Type: research
[ASAP] Synthesis of Artesunic Acid –Coumarin Hybrids as Potential Antimelanoma Agents
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00019 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 24, 2023 Category: Chemistry Authors: Claudio Zippilli, Silvia Filippi, Silvia Cesarini, Bruno Mattia Bizzarri, Pauline Conigliaro, Elisa De Marchi, Lorenzo Botta, and Raffaele Saladino Source Type: research
[ASAP] Synthesis of Veliparib Prodrugs and Determination of Drug-Release-Dependent PARP ‑1 Inhibition
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00065 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 24, 2023 Category: Chemistry Authors: Matteo Borgini and Peter Wipf Source Type: research
[ASAP] Modular One-Pot Strategy for the Synthesis of Heterobivalent Tracers
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00057 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 21, 2023 Category: Chemistry Authors: Thibaud Bailly, Sacha Bodin, Victor Goncalves, Franck Denat, Cle ́ment Morgat, Aurélie Prignon, and Ibai E. Valverde Source Type: research
[ASAP] Cytosolic Enzymes Generate Cannabinoid Metabolites 7 ‑Carboxycannabidiol and 11-Nor-9-carboxytetrahydrocannabinol
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00017 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 20, 2023 Category: Chemistry Authors: Jessica L. Beers, Aurora K. Authement, Nina Isoherranen, and Klarissa D. Jackson Source Type: research
[ASAP] Novel Thienopyrrole Compounds for Treating Autoimmune Diseases and Inflammatory Conditions
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00131 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 20, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Addressing the Osimertinib Resistance Mutation EGFR-L858R/C797S with Reversible Aminopyrimidines
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00514 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 18, 2023 Category: Chemistry Authors: Tobias Grabe, Kirujan Jeyakumar, Janina Niggenaber, Tom Schulz, Sandra Koska, Silke Kleinbo ̈lting, Michael Edmund Beck, Matthias P. Müller, and Daniel Rauh Source Type: research
[ASAP] Discovery of a Novel Series of Potent SHP2 Allosteric Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00059 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 17, 2023 Category: Chemistry Authors: Alessia Petrocchi, Alessandro Grillo, Luca Ferrante, Pietro Randazzo, Adolfo Prandi, Marilenia De Matteo, Costanza Iaccarino, Monica Bisbocci, Antonella Cellucci, Cristina Alli, Martina Nibbio, Vincenzo Pucci, Je ́rôme Amaudrut, Christian Montalbetti, Source Type: research
[ASAP] Rational Design of Highly Potent and Selective Covalent MAP2K7 Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00029 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 17, 2023 Category: Chemistry Authors: Dalton R. Kim, Meghan J. Orr, Ada J. Kwong, Kristine K. Deibler, Hasan H. Munshi, Cory Seth Bridges, Taylor Jie Chen, Xiaoyu Zhang, H. Daniel Lacorazza, and Karl A. Scheidt Source Type: research
[ASAP] Monoacylglycerol Lipase Modulators for Treating Autism Spectrum Disorders
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00121 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 14, 2023 Category: Chemistry Authors: Ram W. Sabnis and Anika R. Sabnis Source Type: research
[ASAP] Correction to “Profiling the Binding Activities of Peptides and Inhibitors to the U2 Auxiliary Factor Homology Motif (UHM) Domains”
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00123 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 14, 2023 Category: Chemistry Authors: Xinrui Yuan, Kathryn L. Howie, Mona Kazemi Sabzvar, Krishnapriya Chinnaswamy, Jeanne A. Stuckey, and Chao-Yie Yang Source Type: research
[ASAP] Targeted Degradation of KRAS < sup > G12D < /sup > as Potential Therapy in Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00111 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 13, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] PROTAC: Harnessing Targeted Chimeras for Selective BCL ‑2 Degradation in Cancer Treatment
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00113 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 13, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] PROTAC Targeted Degradation of IRAK ‑4 as Potential Treatment in Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00112 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 13, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
