[ASAP] APOBEC3A Catalytic Inactivity Mutation Induces Tertiary Structure Destabilization
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00517 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 14, 2023 Category: Chemistry Authors: Katherine F. M. Jones, Mohamed Shehata, Michael A. Carpenter, Rommie E. Amaro, and Daniel A. Harki Source Type: research
[ASAP] Controlling Ibrutinib ’s Conformations about Its Heterobiaryl Axis to Increase BTK Selectivity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00523 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 14, 2023 Category: Chemistry Authors: Sean T. Toenjes, Bahar S. Heydari, Samuel T. Albright, Ramsey Hazin, Maria A. Ortiz, F. Javier Piedrafita, and Jeffrey L. Gustafson Source Type: research
[ASAP] Accelerated Discovery of Macrocyclic CDK2 Inhibitor QR-6401 by Generative Models and Structure-Based Drug Design
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00515 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 8, 2023 Category: Chemistry Authors: Yang Yu, Junhong Huang, Hu He £, Jing Han, Geyan Ye, Tingyang Xu, Xianqiang SunΦ, Xiumei Chen, Xiaoming Ren, Chunlai Li, Huijuan Li, Wei HuangΩ, Yangyang Liu, Xinjuan Wang, Yongzhi Gao, Nianhe Cheng, Na Guo, Xibo Chen, Jianxia Feng, Yuxia Hua, Chong Li Source Type: research
[ASAP] Correction to “Using Imidazo[2,1‑ < italic toggle="yes" > b < /italic > ][1,3,4]thiadiazol Skeleton to Design and Synthesize Novel MNK Inhibitors ”
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00036 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 8, 2023 Category: Chemistry Authors: Xin Jin, Tingting Qiu, Jianling Xie, Xianfeng Wei, Xuemin Wang, Rilei Yu, Christopher Proud, and Tao Jiang Source Type: research
[ASAP] Effective Combination Therapies for the Treatment of HER2 Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00544 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 7, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] Continuous-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00010 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 3, 2023 Category: Chemistry Authors: Antonella Ilenia Alfano, Sveva Pelliccia, Giacomo Rossino, Orazio Chianese, Vincenzo Summa, Simona Collina, and Margherita Brindisi Source Type: research
[ASAP] Working toward a Globally Diverse and Inclusive Community of Medicinal Chemists of the Future
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00533 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 27, 2023 Category: Chemistry Authors: Kelly Chibale(Editor-in-Chief, ACS Medicinal Chemistry Letters) Source Type: research
[ASAP] Passive Membrane Permeability of Sizable Acyclic β‑Hairpin Peptides
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00486 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 27, 2023 Category: Chemistry Authors: Jillene Moxam, Sarah Naylon, Alexis D. Richaud, Guangkuan Zhao, Alberto Padilla, and Ste ́phane P. Roche Source Type: research
[ASAP] Squaramide Tethered Clindamycin, Chloroquine, and Mortiamide Hybrids: Design, Synthesis, and Antimalarial Activity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00531 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 25, 2023 Category: Chemistry Authors: Thomas Tremblay, Catherine Bergeron, Dominic Gagnon, Christopher Be ́rubé, Normand Voyer, Dave Richard, and Denis Giguère Source Type: research
[ASAP] Agrochemical Lessons for Infectious Disease Research: New Resistance Breaking Antifungal Hits against < italic toggle="yes" > Candida auris < /italic >
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00497 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 25, 2023 Category: Chemistry Authors: Christian Winter, Isabella Siepe, Andrew Wise, Alain Dorali, Anthony G. M. Barrett, and Matthias Witschel Source Type: research
[ASAP] Inhibition of HIV ‑1 Protease by a Boronic Acid with High Oxidative Stability
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00464 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 25, 2023 Category: Chemistry Authors: Brian J. Graham, Ian W. Windsor, and Ronald T. Raines Source Type: research
[ASAP] Discovery of Bis-sulfonamides as Novel Inhibitors of Mitochondrial NADH-Quinone Oxidoreductase (Complex I)
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00504 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 24, 2023 Category: Chemistry Authors: Atsuhito Tsuji, Takahiro Masuya, Norihito Arichi, Shinsuke Inuki, Masatoshi Murai, Hideto Miyoshi, and Hiroaki Ohno Source Type: research
[ASAP] Structure-Based Design of Glycosylated Oxytocin Analogues with Improved Selectivity and Antinociceptive Activity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00455 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 24, 2023 Category: Chemistry Authors: Lajos Z. Szabo ́, Parthasadhireddy Tanguturi, Hannah J. Goodman, Sára Sprőber, Chenxi Liu, Fahad Al-Obeidi, Mitchell J. Bartlett, Torsten Falk, Vlad K. Kumirov, M. Leandro Heien, John M. Streicher, and Robin Polt Source Type: research
[ASAP] Call for Papers: Celebrating the 60th Anniversary of the MIKIW Meeting-in-Miniature
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00528 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 23, 2023 Category: Chemistry Authors: Terry W. Moore(ACS Med. Chem. Lett. Topic Editor) Source Type: research
[ASAP] Discovery of Selective Aldehyde Dehydrogenase Inhibitors for the Treatment of Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00543 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - January 23, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
