[ASAP] Prenylated Chrysin Derivatives as Partial PPAR γ Agonists with Adiponectin Secretion-Inducing Activity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00511 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 6, 2023 Category: Chemistry Authors: Seungchan An, Hyejin Ko, Hongjun Jang, In Guk Park, Sungjin Ahn, Seok Young Hwang, Junpyo Gong, Soyeon Oh, Soo Yeon Kwak, Yeonjin Lee, Hyoungsu Kim, and Minsoo Noh Source Type: research

[ASAP] Readily Accessible High-Throughput Experimentation: A General Protocol for the Preparation of ChemBeads and EnzyBeads
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00491 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 3, 2023 Category: Chemistry Authors: Anna C. Impastato, Jesse T. C. Brown, Ying Wang, and Noah P. Tu Source Type: research

[ASAP] Development of Oligomeric Mannose-6-phosphonate Conjugates for Targeted Protein Degradation
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00479 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 3, 2023 Category: Chemistry Authors: Christopher M. Stevens, Yaxian Zhou, Peng Teng, Lauren N. Rault, Yaxian Liao, and Weiping Tang Source Type: research

[ASAP] Conversion of a Cardiac Muscle Modulator from an Inhibitor to an Activator
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00033 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 3, 2023 Category: Chemistry Authors: Fangze Cai, Thomas Kampourakis, Priyanka Parijat, Kieran T. Cockburn, and Brian D. Sykes Source Type: research

[ASAP] Discovery of < bold > CVN636 < /bold > : A Highly Potent, Selective, and CNS Penetrant mGluR < sub > 7 < /sub > Allosteric Agonist
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00529 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 2, 2023 Category: Chemistry Authors: Louise Dickson, Martin Teall, Elodie Chevalier, Toni Cheung, Gemma M. Liwicki, Stephen Mack, Anne Stephenson, Kathryn White, Richard Fosbeary, David C. Harrison, Nicola L. Brice, Kevin Doyle, Roberto Ciccocioppo, Chaobo Wu, Sarah Almond △, Toshal R. Pat Source Type: research

[ASAP] Discovery of Orally Bioavailable FGFR2/FGFR3 Dual Inhibitors via Structure-Guided Scaffold Repurposing Approach
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00003 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 28, 2023 Category: Chemistry Authors: Minh H. Nguyen, Hai-Fen Ye, Yao Xu, Lisa Truong, April Horsey, Peng Zhao, Evan D. Styduhar, Michelle Frascella, Lynn Leffet, Kelly Federowicz, Elham Behshad, Anlai Wang, Ke Zhang, Michael R. Witten, Chao Qi, Ravi Jalluri, Cheng-Tsung Lai, Onur Atasoylu, J Source Type: research

[ASAP] Development of the Inverse Sonogashira Reaction for DEL Synthesis
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00477 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 23, 2023 Category: Chemistry Authors: Ayun Luo, Hongxia Zhou, Qini Hua, Yufang An, Hangke Ma, Xue Zhao, Kexin Yang, and Yun Jin Hu Source Type: research

[ASAP] Contemporary Progress and Opportunities in RNA-Targeted Drug Discovery
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00020 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 23, 2023 Category: Chemistry Authors: Amanda L. Garner Source Type: research

[ASAP] Trust Your Gut: Strategies and Tactics for Intestinally Restricted Drugs
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00001 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 22, 2023 Category: Chemistry Authors: Ruth Dorel, Alice R. Wong, and James J. Crawford Source Type: research

[ASAP] Development and Characterization of Fluorescent Probes for the G Protein-Coupled Receptor 35
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00461 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 22, 2023 Category: Chemistry Authors: Lai Wei, Kaijing Xiang, Hongjian Kang, Yancheng Yu, Hongjie Fan, Han Zhou, Tao Hou, Yonglin Ge, Jixia Wang, Zhimou Guo, Yang Chen, Yaopeng Zhao, and Xinmiao Liang Source Type: research

[ASAP] Structural Study of Potent Triazole-Based Inhibitors of < named-content content-type="genus-species" xlink:type="simple" > Staphylococcus aureus < /named-content > Biotin Protein Ligase
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00505 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 21, 2023 Category: Chemistry Authors: Damian L. Stachura, Stephanie Nguyen, Steven W. Polyak, Blagojce Jovcevski, John B. Bruning, and Andrew D. Abell Source Type: research

[ASAP] Introducing Conformational Restraints on 25CN-NBOH: A Selective 5 ‑HT < sub > 2A < /sub > Receptor Agonist
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00014 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 20, 2023 Category: Chemistry Authors: Emil Marcher-Rrsted, Jitka Nykodemova ́, Kasper Harpse, Anders A. Jensen, and Jesper L. Kristensen Source Type: research

[ASAP] Ligand Screening System for the RXR α Heterodimer Using the Fluorescence RXR Agonist CU-6PMN
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00509 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 20, 2023 Category: Chemistry Authors: Mayu Kawasaki, Tomoharu Motoyama, Shoya Yamada, Masaki Watanabe, Michiko Fujihara, Akira Kambe, Shogo Nakano, Hiroki Kakuta, and Sohei Ito Source Type: research

[ASAP] Recent Advances in Alchemical Binding Free Energy Calculations for Drug Discovery
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00541 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 16, 2023 Category: Chemistry Authors: Ingo Muegge and Yuan Hu Source Type: research

[ASAP] Pyridine-Based 1,2,4-Triazolo-Tethered Indole Conjugates Potentially Affecting TNKS and PI3K in Colorectal Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00475 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - February 16, 2023 Category: Chemistry Authors: Prasanna A. Yakkala, Samir R. Panda, Vegi G. M. Naidu, Syed Shafi, and Ahmed Kamal Source Type: research