[ASAP] Aroylhydrazone Glycoconjugate Prochelators Exploit Glucose Transporter 1 (GLUT1) to Target Iron in Cancer Cells
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00250 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 18, 2022 Category: Chemistry Authors: Yu-Shien Sung, Baris Kerimoglu, Aikseng Ooi, and Elisa Tomat Source Type: research
[ASAP] Fragment Ligands of the m < sup > 6 < /sup > A ‑RNA Reader YTHDF2
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00303 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 17, 2022 Category: Chemistry Authors: Francesco Nai, Raed Nachawati, Frantis ̌ek Zálešák, Xiang Wang, Yaozong Li, and Amedeo Caflisch Source Type: research
[ASAP] 2 ‑Amino-1,3,4-thiadiazoles as Glutaminyl Cyclases Inhibitors Increase Phagocytosis through Modification of CD47-SIRPα Checkpoint
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00256 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 16, 2022 Category: Chemistry Authors: Eunsun Park, Kyung-Hee Song, Darong Kim, Minyoung Lee, Nguyen Van Manh, Hee Kim, Ki Bum Hong, Jeewoo Lee, Jie-Young Song, and Soosung Kang Source Type: research
[ASAP] Triazine-Based Covalent DNA-Encoded Libraries for Discovery of Covalent Inhibitors of Target Proteins
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00127 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 15, 2022 Category: Chemistry Authors: Linjie Li, Mingbo Su, Weiwei Lu, Hongzhi Song, Jiaxiang Liu, Xin Wen, Yanrui Suo, Jingjing Qi, Xiaomin Luo, Yu-Bo Zhou, Xin-Hua Liao, Jia Li, and Xiaojie Lu Source Type: research
[ASAP] Turning the Other Cheek: Influence of the < italic toggle="yes" > cis < /italic > -Tetrafluorocyclohexyl Motif on Physicochemical and Metabolic Properties
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00312 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 14, 2022 Category: Chemistry Authors: Yong Wang, Wendy Lee, Yi-Chen Chen, Yuhui Zhou, Emile Plise, Madyson Migliozzi, and James J. Crawford Source Type: research
[ASAP] Novel Bcl ‑2 Inhibitors Selectively Disrupt the Autophagy-Specific Bcl-2–Beclin 1 Protein–Protein Interaction
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00309 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 12, 2022 Category: Chemistry Authors: Xiaonan Dong, Qiren Liang, Yun-Zu Pan, Xiaoyu Wang, Yi-Chun Kuo, Wei-Chung Chiang, Xuewu Zhang, Noelle S. Williams, Josep Rizo, Beth Levine, and Jef K. De Brabander Source Type: research
[ASAP] Multicomponent Macrocyclic IL-17a Modifier
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00257 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 12, 2022 Category: Chemistry Authors: Eman Abdelraheem, Max Lubberink, Wenja Wang, Jingyao Li, Atilio Reyes Romero, Robin van der Straat, Xiaochen Du, Matthew Groves, and Alexander Do ̈mling Source Type: research
[ASAP] Novel 3 ‑Aminopyrrolidine and Piperidine Macrocyclic Orexin Receptor Agonists for Treating Sleep Disorders
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00341 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 12, 2022 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Identification of α‑Synuclein Proaggregator: Rapid Synthesis and Streamlining RT-QuIC Assays in Parkinson’s Disease
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00138 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 11, 2022 Category: Chemistry Authors: Fumito Takada, Takahito Kasahara, Kentaro Otake, Takamitsu Maru, Masanori Miwa, Kei Muto, Minoru Sasaki, Yoshihiko Hirozane, Masato Yoshikawa, and Junichiro Yamaguchi Source Type: research
[ASAP] Decarboxylative Cross-Coupling: A Radical Tool in Medicinal Chemistry
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00286 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 10, 2022 Category: Chemistry Authors: Gabriele Laudadio, Maximilian D. Palkowitz, Tamara El-Hayek Ewing, and Phil S. Baran Source Type: research
[ASAP] Pyrimido[5,4 ‑ < italic toggle="yes" > d < /italic > ]pyrimidine-Based Compounds as a Novel Class of Antitrypanosomal and Antileishmanial Agents
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00170 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 9, 2022 Category: Chemistry Authors: Andre ́ Lopes, Nuno Santarém, Anabela Cordeiro-da-Silva, and M. Alice Carvalho Source Type: research
[ASAP] Novel Coronavirus Main Protease Di- and Tripeptide Inhibitors for Treating COVID-19
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00332 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 8, 2022 Category: Chemistry Authors: C. S. Brian Chia and Yi Yang See Source Type: research
[ASAP] Substituted 6,7-Dihydro ‑5 < italic toggle="yes" > H < /italic > ‑Benzo[7]annulene Compounds as Selective Estrogen Receptor Degraders for Treating Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00342 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 4, 2022 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Identification of a BAZ2A-Bromodomain Hit Compound by Fragment Growing
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00173 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 3, 2022 Category: Chemistry Authors: Andrea Dalle Vedove, Giulia Cazzanelli, Laurent Batiste, Jean-Re ́my Marchand, Dimitrios Spiliotopoulos, Jessica Corsi, Vito Giuseppe D’Agostino, Amedeo Caflisch, and Graziano Lolli Source Type: research
[ASAP] Discovery of Novel 2 ‑Carbamoyl Morpholine Derivatives as Highly Potent and Orally Active Direct Renin Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00280 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - August 1, 2022 Category: Chemistry Authors: Daisuke Iijima, Hiroshi Sugama, Nobumasa Awai, Yoichi Takahashi, Yuko Togashi, Tohru Takebe, Jianshu Xie, Jingkang Shen, Ying Ke, Hidenori Akatsuka, Takayuki Kawaguchi, Kei Takedomi, Akiko Kashima, Masashi Nishio, Yosuke Inui, Hikaru Yoneda, Guangxin Xia, Source Type: research
