[ASAP] Quantum Annealing Designs Nonhemolytic Antimicrobial Peptides in a Discrete Latent Space
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00487 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 13, 2023 Category: Chemistry Authors: Andrejs Tuc ̌s, Francois Berenger, Akiko Yumoto, Ryo Tamura, Takanori Uzawa, and Koji Tsuda Source Type: research
[ASAP] Photo-Flow Technology for Chemical Rearrangements: A Powerful Tool to Generate Pharmaceutically Relevant Compounds
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00072 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 12, 2023 Category: Chemistry Authors: Antonella Ilenia Alfano, Sveva Pelliccia, Giacomo Rossino, Orazio Chianese, Vincenzo Summa, Simona Collina, and Margherita Brindisi Source Type: research
[ASAP] Novel AHR Agonists for Treating Psoriasis
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00120 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 12, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] 1,2,4-Triazine Derivatives as NLRP3 Inhibitors for Treating Diseases
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00122 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 12, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Discovery of First-in-Class Small Molecule Inhibitors of Lymphocyte Activation Gene 3 (LAG-3)
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00054 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 11, 2023 Category: Chemistry Authors: Somaya A. Abdel-Rahman, Ashfaq Ur Rehman, and Moustafa T. Gabr Source Type: research
[ASAP] Inhibition of Thiamine Diphosphate-Dependent Enzymes by Triazole-Based Thiamine Analogues
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00047 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 11, 2023 Category: Chemistry Authors: Alex H. Y. Chan, Terence C. S. Ho, Imam Fathoni, Rebecca Pope, Kevin J. Saliba, and Finian J. Leeper Source Type: research
[ASAP] Selective Wee1 Inhibitors Led to Antitumor Activity < italic toggle="yes" > In Vitro < /italic > and Correlated with Myelosuppression
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00481 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 7, 2023 Category: Chemistry Authors: Satenig Guler, Maria C. DiPoto, Alejandro Crespo, Richard Caldwell, Benjamin Doerfel, Nina Grossmann, Kevin Ho, Bayard Huck, Christopher CV Jones, Ruoxi Lan, Djordje Musil, Justin Potnick, Heike Schilke, Brian Sherer, Stephanie Simon, Christian Sirrenberg Source Type: research
[ASAP] Methyl and Fluorine Effects in Novel Orally Bioavailable Keap1 –Nrf2 PPI Inhibitor
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00067 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 7, 2023 Category: Chemistry Authors: Kazuki Otake, Minoru Ubukata, Noboru Nagahashi, Naoki Ogawa, Yoshiji Hantani, Rie Hantani, Tsuyoshi Adachi, Akihiro Nomura, Keishi Yamaguchi, Mariko Maekawa, Hideaki Mamada, Takahisa Motomura, Motohide Sato, and Kazuhito Harada Source Type: research
[ASAP] Artefenomel Regioisomer RLA-3107 Is a Promising Lead for the Discovery of Next-Generation Endoperoxide Antimalarials
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00039 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - April 4, 2023 Category: Chemistry Authors: Brian R. Blank, Jiri Gut, Philip J. Rosenthal, and Adam R. Renslo Source Type: research
[ASAP] An Isomer of Galidesivir That Potently Inhibits Influenza Viruses and Members of the < italic toggle="yes" > Bunyavirales < /italic > Order
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00048 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 30, 2023 Category: Chemistry Authors: Kevin J. Sparrow, Rinu Shrestha, James M. Wood, Keith Clinch, Brett L. Hurst, Hong Wang, Brian B. Gowen, Justin G. Julander, E. Bart Tarbet, Alice M. McSweeney Ψ, Vernon K. WardΨ, Gary B. Evans, and Lawrence. D. Harris Source Type: research
[ASAP] Anagrelide: A Clinically Effective cAMP Phosphodiesterase 3A Inhibitor with Molecular Glue Properties
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00092 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 28, 2023 Category: Chemistry Authors: Nicholas A. Meanwell Source Type: research
[ASAP] Using Transcriptomics and Cell Morphology Data in Drug Discovery: The Long Road to Practice
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00015 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 22, 2023 Category: Chemistry Authors: Lavinia-Lorena Pruteanu and Andreas Bender Source Type: research
[ASAP] Evaluation of 1,3,4-Thiadiazole Carbonic Anhydrase Inhibitors for Gut Decolonization of Vancomycin-Resistant Enterococci
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00032 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 21, 2023 Category: Chemistry Authors: Nader S. Abutaleb, Annadka Shrinidhi, Aloka B. Bandara, Mohamed N. Seleem, and Daniel P. Flaherty Source Type: research
[ASAP] Profiling the Binding Activities of Peptides and Inhibitors to the U2 Auxiliary Factor Homology Motif (UHM) Domains
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00537 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 21, 2023 Category: Chemistry Authors: Xinrui Yuan, Kathryn L. Howie, Mona Kazemi Sabzvar, Krishnapriya Chinnaswamy, Jeanne A. Stuckey, and Chao-Yie Yang Source Type: research
[ASAP] Discovery and Optimization of a Novel Macrocyclic Amidinourea Series Active as Acidic Mammalian Chitinase Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00472 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - March 21, 2023 Category: Chemistry Authors: Lorenzo Jacopo Ilic Balestri, Claudia Immacolata Trivisani, Francesco Orofino, Diego Fiorucci, Giuseppina Ivana Truglio, Ilaria D ’Agostino, Federica Poggialini, Lorenzo Botta, Jean-Denis Docquier, and Elena Dreassi Source Type: research
