[ASAP] Nitrogen-Containing 2,3-Dihydroquinazolinone Compounds as Na < sub > v < /sub > 1.8 Inhibitors for Treating Pain and Cardiovascular Diseases
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00235 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Examination of the Impact of Triazole Position within Linkers on Solubility and Lipophilicity of a CDK9 Degrader Series
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00082 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Oluwatosin R. Ayinde, Chia Sharpe, Emily Stahl, Robert J. Tokarski II, James R. Lerma, Natarajan Muthusamy, John C. Byrd, and James R. Fuchs Source Type: research
[ASAP] < italic toggle="yes" > N < /italic > ‑Alkyl Carbamoylimidazoles as Versatile Synthons for the Synthesis of Urea-Based PSMA Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00087 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Narendar Reddy Gade, Jatinder Kaur, Atul Bhardwaj, Edris Ebrahimi, Jennifer Dufour, Melinda Wuest, and Frank Wuest Source Type: research
[ASAP] Microbiome –Gut–Brain Axis Modulation: New Approaches in Treatment of Parkinson’s Disease and Amyotrophic Lateral Sclerosis
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00221 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] Subhallucinogenic Concentrations of Substituted Phenethylamines as a Novel Therapeutic Approach for Inflammatory and Neurological Disorders
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00220 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] Unveiling New KRAS < sup > G12D < /sup > Inhibitors: A Promising Approach for Pancreatic Cancer Therapy
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00222 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 9, 2023 Category: Chemistry Authors: Robert B. Kargbo Source Type: research
[ASAP] Fused Bicyclic Heteroaryl Compounds as NLRP3 Inhibitors for Treating Asthma or COPD
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00236 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 6, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
[ASAP] Virtual Special Issue: New Drug Modalities in Medicinal Chemistry, Pharmacology, and Translational Science
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00147 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 6, 2023 Category: Chemistry Authors: Jeffrey Aube ́(Associate Editor, ACS Medicinal Chemistry Letters), Craig W. Lindsley(Editor-in-Chief, Journal of Medicinal Chemistry), and Christa E. Müller(Editor-in-Chief, ACS Pharmacology & Translational Science) Source Type: research
[ASAP] Discovery of New Binders for DCAF1, an Emerging Ligase Target in the Targeted Protein Degradation Field
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00104 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 2, 2023 Category: Chemistry Authors: Anna Vulpetti, Philipp Holzer, Niko Schmiedeberg, Patricia Imbach-Weese, Carole Pissot-Soldermann, Gregory J. Hollingworth, Thomas Radimerski, Claudio R. Thoma, Therese-Marie Stachyra, Matthias Wojtynek, Magdalena Maschlej, Suzanne Chau, Ansgar Schuffenha Source Type: research
[ASAP] High-Throughput Purification in Drug Discovery: Scaling New Heights of Productivity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00073 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 31, 2023 Category: Chemistry Authors: Mark Jones and Ross L. Goodyear Source Type: research
[ASAP] TMPRSS2 Inhibitor Discovery Facilitated through an < italic toggle="yes" > In Silico < /italic > and Biochemical Screening Platform
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00035 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 30, 2023 Category: Chemistry Authors: Amanda L. Peiffer, Julie M. Garlick, Yujin Wu, Jesse W. Wotring, Sahil Arora, Alexander S. Harmata, Daniel A. Bochar, Corey J. Stephenson, Matthew B. Soellner, Jonathan Z. Sexton, Charles L. Brooks, III, and Anna K. Mapp Source Type: research
[ASAP] Novel Concept for Super-Soft Topical Drugs: Deactivation by an Enzyme-Induced Switch into an Inactive Conformation
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00169 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 30, 2023 Category: Chemistry Authors: Gebhard Thoma, Eric Vangrevelinghe, Alexandre Luneau, Philippe Piechon, Christian Beerli, and Hans-Guenter Zerwes Source Type: research
[ASAP] Design and Synthesis of Pyrazole-Based Macrocyclic Kinase Inhibitors Targeting BMPR2
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00127 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 30, 2023 Category: Chemistry Authors: Jennifer A. Amrhein, Guiqun Wang, Benedict-Tilman Berger, Lena M. Berger, Amalia D. Kalampaliki, Andreas Kra ̈mer, Stefan Knapp, and Thomas Hanke Source Type: research
[ASAP] Recent Developments in Mass Spectrometry to Support Next-Generation Synthesis and Screening
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00040 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 30, 2023 Category: Chemistry Authors: Nari N. Talaty, Robert W. Johnson, James Sawicki, Omprakash Nacham, and Stevan W. Djuric Source Type: research
[ASAP] Novel Quinoline Compounds as KRAS Inhibitors for Treating Cancer
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.3c00195 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - May 26, 2023 Category: Chemistry Authors: Ram W. Sabnis Source Type: research
