[ASAP] Novel Macrocyclic 1,3,4-Oxadiazoles as CFTR Modulators for Treating Cystic Fibrosis
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00288 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 30, 2022 Category: Chemistry Authors: Ram W. Sabnis Source Type: research

[ASAP] Novel Isoindolinone-Based Analogs of the Natural Cyclic Peptide Fenestin A: Synthesis and Antitumor Activity
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00149 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 29, 2022 Category: Chemistry Authors: Huanli Zhang, Jingwan Wu, Jingchun Wang, Shimei Xiao, Lei Zhao, Rui Yan, Xiaodan Wu, Zhiqiang Wang, Li Fan, and Yingxue Jin Source Type: research

[ASAP] Discovery of Antibacterial Contezolid Acefosamil: Innovative < italic toggle="yes" > O < /italic > ‑Acyl Phosphoramidate Prodrug for IV and Oral Therapies
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00191 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 29, 2022 Category: Chemistry Authors: Jinqian Liu, Wen Wang, Changqing Wang, Li Zhang, Xueliang Zhang, Shicong Liu, Yunhua Xu, Hailin Wang, Qing Dai, Chun Liu, Xinghai Wang, Zhengyu Yuan, and Mikhail F. Gordeev Source Type: research

[ASAP] Discovery of Benzylpiperazine Derivatives as CNS-Penetrant and Selective Histone Deacetylase 6 Inhibitors
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00081 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 28, 2022 Category: Chemistry Authors: Kosuke Hashimoto, Soichiro Ide, Mayumi Arata, Akiko Nakata, Akihiro Ito, Takashi K. Ito, Norio Kudo, Bangzhong Lin, Kazuto Nunomura, Keiko Tsuganezawa ≡, Minoru YoshidaΠ, Yasuo Nagaoka, and Takaaki Sumiyoshi Source Type: research

[ASAP] Nanoacetylated < italic toggle="yes" > N < /italic > ‑(4-Hydroxyphenyl) Retinamide Modulates Histone Acetylation–Methylation Epigenetic Disparity to Restrict Epithelial–Mesenchymal Transition in Neuroblastoma
ACS Medicinal Chemistry LettersDOI: 10.1021/acsmedchemlett.2c00135 (Source: ACS Medicinal Chemistry Letters)
Source: ACS Medicinal Chemistry Letters - June 27, 2022 Category: Chemistry Authors: Atul Dev, Mohammed Nadim Sardoiwala, Angela Sharma, Soni Jignesh MohanBhai, Surajit Karmakar, and Subhasree Roy Choudhury Source Type: research