[ASAP] Design and Characterization of Squaramic Acid-Based Prostate-Specific Membrane Antigen Inhibitors for Prostate Cancer
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00309 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 10, 2023 Category: Chemistry Authors: Xinlin Wang, Yimin Chen, Yuqing Xiong, Longfei Zhang, Beibei Wang, Yajun Liu, and Mengchao Cui Source Type: research
[ASAP] Development of a Suite of Gadolinium-Free OATP1-Targeted Paramagnetic Probes for Liver MRI
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.2c01561 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 9, 2023 Category: Chemistry Authors: Sean W. McRae, Michael Cleary, Daniel DeRoche, Francisco M. Martinez, Ying Xia, Peter Caravan, Eric M. Gale, John A. Ronald, and Timothy J. Scholl Source Type: research
[ASAP] Discovery and Optimization of Novel Biphenyl Derivatives Bearing Cyclopropyl Linkage as Potent Programmed Cell Death-1/Programmed Cell Death-Ligand 1 Inhibitors
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00205 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 9, 2023 Category: Chemistry Authors: Tongfei Jing, Zhijing Zhang, Zhenghui Kang, Jianshan Mo, Xiaotong Yue, Ziyou Lin, Xiang Fu, Chang Liu, Hang Ma, Xiaolei Zhang, and Wenhao Hu Source Type: research
[ASAP] Quinazoline-2-Carboxamides as Selective PET Radiotracers for Matrix Metalloproteinase-13 Imaging in Atherosclerosis
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.2c02107 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 9, 2023 Category: Chemistry Authors: Ariel Buchler, Uzair S. Ismailani, Nicole MacMullin, Faduma Abdirahman, Myriam Adi, Christina Bi, Catherine Jany, Jeffrey W. Keillor, and Benjamin H. Rotstein Source Type: research
[ASAP] < sup > 68 < /sup > Ga-Labeled TMTP1 Derivatives with Moderate Hydrophilicity for Positron Emission Tomography of Hepatocellular Carcinoma in High Contrast
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00111 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 9, 2023 Category: Chemistry Authors: Xiaowei Fan, Xiaoxiao Wang, Zijing Li, and Yesen Li Source Type: research
[ASAP] Stereochemical Control of Splice Modulation in FD-895 Analogues
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.2c01893 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Warren C. Chan, Kelsey A. Trieger, James J. La Clair, Catriona H. M. Jamieson, and Michael D. Burkart Source Type: research
[ASAP] Correction to “Discovery of Nanomolar Melanocortin‑3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High Throughput ‘Unbiased’ Screening Campaign”
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00588 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Skye R. Doering, Katie Freeman, Ginamarie Debevec, Phaedra Geer, Radleigh G. Santos, Travis M. Lavoi, Marc A. Giulianotti, Clemencia Pinilla, Jon R. Appel, Richard A. Houghten, Mark D. Ericson, and Carrie Haskell-Luevano Source Type: research
[ASAP] First-in-Class Selective Inhibitors of the Lysine Acetyltransferase KAT8
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.2c01937 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Francesco Fiorentino, Sara Sementilli, Martina Menna, Federica Turrisi, Stefano Tomassi, Francesca Romana Pellegrini, Angela Iuzzolino, Francesca D ’Acunzo, Alessandra Feoli, Hannah Wapenaar, Sophie Taraglio, Caterina Fraschetti, Donatella Del Bufalo, G Source Type: research
[ASAP] Discovery of Norisoboldine Analogue III < sub > 11 < /sub > as a Novel and Potent Aryl Hydrocarbon Receptor Agonist for the Treatment of Ulcerative Colitis
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00287 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Li Lin, Yongmin Liu, Li Chen, Yue Dai, and Yufeng Xia Source Type: research
[ASAP] < italic toggle="yes" > In Vitro < /italic > and < italic toggle="yes" > In Vivo < /italic > Evaluation of ABCG2 (BCRP) Inhibitors Derived from Ko143
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00168 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Melanie Zechner, Claudia A. Castro Jaramillo, Nadine S. Zubler, Marco F. Taddio, Linjing Mu, Karl-Heinz Altmann, and Stefanie D. Kra ̈mer Source Type: research
[ASAP] Trioxacarcin A Interactions with G ‑Quadruplex DNA Reveal Its Potential New Targets as an Anticancer Agent
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00178 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Shaowen Yin, Wenxian Lan, Xianfeng Hou, Zhijun Liu, Hongjuan Xue, Chunxi Wang, Gong-Li Tang, and Chunyang Cao Source Type: research
[ASAP] Discovery of PMSA Derivative < bold > 11 < /bold > as a Novel Lead Compound for Therapeutic Treatment of Osteoporosis < italic toggle="yes" > In Vitro < /italic > and < italic toggle="yes" > In Vivo < /italic >
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00114 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 8, 2023 Category: Chemistry Authors: Zhihao Chen, Karthik Rajan Rajamanickam, Mina Ding, Sang Kyoon Kim, Sang-wook Park, Eunae Kim, Sunwoo Lee, and Tae-Hoon Lee Source Type: research
[ASAP] A Molecular Toolbox of Positron Emission Tomography Tracers for General Anesthesia Mechanism Research
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.2c01965 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 5, 2023 Category: Chemistry Authors: Xiaoxiao Wang, Tao Wang, Xiaowei Fan, Zhao Zhang, Yingwei Wang, and Zijing Li Source Type: research
[ASAP] X ‑ray Crystal Structure-Guided Discovery of Novel Indole Analogues as Colchicine-Binding Site Tubulin Inhibitors with Immune-Potentiating and Antitumor Effects against Melanoma
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00011 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 5, 2023 Category: Chemistry Authors: Yichang Ren, Yuxi Wang, Jin Liu, Ting Liu, Lin Yuan, Chengyong Wu, Zichao Yang, and Jianjun Chen Source Type: research
[ASAP] Rationally Engineered CYP3A4 Fluorogenic Substrates for Functional Imaging Analysis and Drug –Drug Interaction Studies
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00101 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 5, 2023 Category: Chemistry Authors: Rong-Jing He, Zhen-Hao Tian, Jian Huang, Meng-Ru Sun, Feng Wei, Chun-Yu Li, Hai-Rong Zeng, Feng Zhang, Xiao-Qing Guan, Yan Feng, Xiang-Ming Meng, Hui Yang, and Guang-Bo Ge Source Type: research
