[ASAP] Targeting MET: Discovery of Small Molecule Inhibitors as Non-Small Cell Lung Cancer Therapy
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00028 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - June 1, 2023 Category: Chemistry Authors: Chaofan Wang δ and Xiaoyun Luδ Source Type: research

[ASAP] Computational Design, Synthesis, and Biological Evaluation of Diimidazole Analogues Endowed with Dual PCSK9/HMG-CoAR-Inhibiting Activity
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00279 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - June 1, 2023 Category: Chemistry Authors: Carmen Lammi, Enrico M. A. Fassi, Marco Manenti, Marta Brambilla, Maria Conti, Jianqiang Li, Gabriella Roda, Marina Camera, Alessandra Silvani, and Giovanni Grazioso Source Type: research

[ASAP] Characterization of a Potent and Orally Bioavailable Lys-Covalent Inhibitor of Apoptosis Protein (IAP) Antagonist
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00467 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - June 1, 2023 Category: Chemistry Authors: Parima Udompholkul, Ana Garza-Granados, Giulia Alboreggia, Carlo Baggio, Jack McGuire, Scott D. Pegan, and Maurizio Pellecchia Source Type: research

[ASAP] Redirection of CAR ‑T Cell Cytotoxicity Using Metabolic Glycan Labeling with Unnatural Sugars
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00048 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - June 1, 2023 Category: Chemistry Authors: Jeong Hyeon Cha, Eunsu Kim, Hyeong Ji Lee, Young-Ho Lee, Jeonghyun Lee, Eunha Kim, and Chan Hyuk Kim Source Type: research

[ASAP] Targeting Pancreatic Cancer with Novel Plumbagin Derivatives: Design, Synthesis, Molecular Mechanism, < italic toggle="yes" > In Vitro < /italic > and < italic toggle="yes" > In Vivo < /italic > Evaluation
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00394 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 31, 2023 Category: Chemistry Authors: Suresh Awale, Hayato Baba, Nguyen Duy Phan, Min Jo Kim, Juthamart Maneenet, Koichi Sawaki, Mitsuro Kanda, Tomoyuki Okumura, Tsutomu Fujii, Takuya Okada, Takahiro Maruyama, Takahiro Okada, and Naoki Toyooka Source Type: research

[ASAP] Escaping from Flatland: Multiparameter Optimization Leads to the Discovery of Novel Tetrahydropyrido[4,3 ‑ < italic toggle="yes" > d < /italic > ]pyrimidine Derivatives as Human Immunodeficiency Virus ‑1 Non-nucleoside Reverse Transcriptase Inhibitors with Superior Antiviral Activities against Non-nucleoside Reverse Transcriptase Inhibitor-Resistant Variants and Favorable Drug-like Profiles
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00275 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 31, 2023 Category: Chemistry Authors: Zhao Wang, Prem Prakash Sharma, Brijesh Rathi, Minghui Xie, Erik De Clercq, Christophe Pannecouque, Dongwei Kang, Peng Zhan, and Xinyong Liu Source Type: research

[ASAP] < italic toggle="yes" > De Novo < /italic > Design of Nurr1 Agonists < italic toggle="yes" > via < /italic > Fragment-Augmented Generative Deep Learning in Low-Data Regime
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00485 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 31, 2023 Category: Chemistry Authors: Marco Ballarotto, Sabine Willems, Tanja Stiller, Felix Nawa, Julian A. Marschner, Francesca Grisoni, and Daniel Merk Source Type: research

[ASAP] Fragment-Based Discovery of Azocyclic Alkyl Naphthalenesulfonamides as Keap1-Nrf2 Inhibitors for Acute Lung Injury Treatment
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00686 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 31, 2023 Category: Chemistry Authors: Jianyu Yan, Yue Li, Li Ding, Ruilin Hou, Chengguo Xing, Chengshi Jiang, Zhenyuan Miao, and Chunlin Zhuang Source Type: research

[ASAP] Correction to “Advances in Epilepsy: Mechanisms, Clinical Trials, and Drug Therapies”
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00843 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 30, 2023 Category: Chemistry Authors: Tingting Hu, Jifa Zhang, Jiaxing Wang, Leihao Sha, Yilin Xia, Tyler C. Ortyl, Xiaohe Tian, and Lei Chen Source Type: research

[ASAP] [ < sup > 68 < /sup > Ga]Ga-Ornibactin for < named-content content-type="genus-species" xlink:type="simple" > Burkholderia cepacia < /named-content > complex Infection Imaging Using Positron Emission Tomography
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00469 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 30, 2023 Category: Chemistry Authors: Katerina Bendova, Vladislav Raclavsky, Radko Novotny, Dominika Luptakova, Miroslav Popper, Zbynek Novy, Marian Hajduch, and Milos Petrik Source Type: research

[ASAP] Design and Synthesis of Bouchardatine Derivatives as a Novel AMP-Activated Protein Kinase Activator for the Treatment of Colorectal Cancer
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00085 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 30, 2023 Category: Chemistry Authors: Yao-Hao Xu, Yu-Tao Hu, Shu-Min Xu, Bing-Bing Song, Hao Yuan, Dan-Dan Zhao, Shi-Yao Guo, Zhi Jiang, Li-Yuan Wei, Yong Rao, Jia-Heng Tan, Shi-Liang Huang, Qing-Jiang Li, Shuo-Bin Chen, and Zhi-Shu Huang Source Type: research

[ASAP] PINK1-Dependent Mitophagy Inhibits Elevated Ubiquitin Phosphorylation Caused by Mitochondrial Damage
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00555 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 30, 2023 Category: Chemistry Authors: Olivia A. Lambourne, Shane Bell, Le ́a P. Wilhelm, Erika B. Yarbrough, Gabriel G. Holly, Oliver M. Russell, Arwa M. Alghamdi, Azeza M. Fdel, Carmine Varricchio, Emma L. Lane, Ian G. Ganley, Arwyn T. Jones, Matthew S. Goldberg, and Youcef Mehellou Source Type: research

[ASAP] Visual and Electrochemical Detection of let-7a: A Tumor Suppressor and Biomarker
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00499 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 29, 2023 Category: Chemistry Authors: Zhen Song, Qiang-Yan Zhang, Jia-Jing Li, Jing-Lian Su, Yuan-Hua Liu, Gong-Jun Yang, and Huai-Song Wang Source Type: research

[ASAP] Nonpeptidic Oxazole-Based Prolyl Oligopeptidase Ligands with Disease-Modifying Effects on α‑Synuclein Mouse Models of Parkinson’s Disease
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00235 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 29, 2023 Category: Chemistry Authors: Tommi P. Kilpela ̈inen, Henri T. Pätsi, Reinis Svarcbahs, Ulrika H. Julku, Tony S. Eteläinen, Hengjing Cui, Samuli Auno, Nina Sipari, Susanna Norrbacka, Teppo O. Leino, Maria Jäntti, Timo T. Myöhänen, and Erik A. A. Wallén Source Type: research

[ASAP] Development of a Novel HER2-Targeted Peptide Probe for Dual-Modal Imaging of Tumors
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00347 (Source: Journal of Medicinal Chemistry)
Source: Journal of Medicinal Chemistry - May 29, 2023 Category: Chemistry Authors: Rui Cao, Renda Li, Chaoquan Lai, Hui Shi, Hongguang Liu, and Zhen Cheng Source Type: research