New frontiers in the design and discovery of therapeutics that target calcium ion signaling: a novel approach in the fight against cancer
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 1, 2023 Category: Drugs & Pharmacology Authors: Jyoti Singh Abha Meena Suaib Luqman Source Type: research

Applications of machine learning in microbial natural product drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 31, 2023 Category: Drugs & Pharmacology Authors: Autumn Arnold Jeremie Alexander Gary Liu Jonathan M. Stokes Source Type: research

Optimizing drug discovery using multitasking models for quantitative structure –biological effect relationships: an update of the literature
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 28, 2023 Category: Drugs & Pharmacology Authors: Valeria V. Kleandrova M. Nat ália D. S. Cordeiro Alejandro Speck-Planche Source Type: research

Preclinical discovery and development of nirmatrelvir/ritonavir combinational therapy for the treatment of COVID-19 and the lessons learned from SARS-COV-2 variants
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 24, 2023 Category: Drugs & Pharmacology Authors: Pasquale Pagliano Annamaria Spera Carmine Sellitto Giuliana Scarpati Veronica Folliero Ornella Piazza Gianluigi Franci Valeria Conti Tiziana Ascione Source Type: research

Exploring the current use of animal models in glaucoma drug discovery: where are we in 2023?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 23, 2023 Category: Drugs & Pharmacology Authors: Renu Agarwal Puneet Agarwal Igor Iezhitsa Source Type: research

The current role and evolution of X-ray crystallography in drug discovery and development
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 18, 2023 Category: Drugs & Pharmacology Authors: Vanessa Bijak Michal Szczygiel Joanna Lenkiewicz Michal Gucwa David R. Cooper Krzysztof Murzyn Wladek Minor Source Type: research

Developing our knowledge of the quinolone scaffold and its value to anticancer drug design
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 18, 2023 Category: Drugs & Pharmacology Authors: Yogesh Singh Neha Bhatia Avadh Biharee Swanand Kulkarni Suresh Thareja Vikramdeep Monga Source Type: research

The preclinical discovery and development of deucravacitinib for the treatment of psoriasis
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 14, 2023 Category: Drugs & Pharmacology Authors: Giulia Coscarella Dalma Malvaso Maria Mannino Giacomo Caldarola Barbara Fossati Clara De Simone Andrea Chiricozzi Ketty Peris Source Type: research

Structural and functional annotation of solute carrier transporters: implication for drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 11, 2023 Category: Drugs & Pharmacology Authors: Vojtech Dvorak Giulio Superti-Furga Source Type: research

Understanding the role of cGAS-STING signaling in ischemic stroke: a new avenue for drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 11, 2023 Category: Drugs & Pharmacology Authors: Chandan Chauhan Ravinder Kumar Kaundal Source Type: research

Opportunities and challenges in new HIV therapeutic discovery: what is the next step?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 10, 2023 Category: Drugs & Pharmacology Authors: Shujing Xu Lin Sun Xinyong Liu Peng Zhan Source Type: research

Recent advances in measurement of metabolic clearance, metabolite profile and reaction phenotyping of low clearance compounds
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 1, 2023 Category: Drugs & Pharmacology Authors: Li Di Source Type: research

Prudent tactics to sail the boat of PARP inhibitors as therapeutics for diverse malignancies
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 1, 2023 Category: Drugs & Pharmacology Authors: Mandeep Rana Amandeep Thakur Charanjit Kaur Chun-Hsu Pan Sung-Bau Lee Jing Ping Liou Kunal Nepali Source Type: research

The premise of capsid assembly modulators towards eliminating HBV persistence
Volume 18, Issue 9, July - December 2023, Page 1031-1041 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 31, 2023 Category: Drugs & Pharmacology Authors: Leda Bassit Franck Amblard Dharmeshkumar Patel Nicolas Biteau Zhe Chen Mahesh Kasthuri Shaoman Zhou Raymond F. Schinazi Source Type: research

Drug design strategies that aim to improve the low solubility and poor bioavailability conundrum in quercetin derivatives
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 29, 2023 Category: Drugs & Pharmacology Authors: Seyedeh Roya Alizadeh Niloofar Savadkouhi Mohammad Ali Ebrahimzadeh Source Type: research