Redirecting the revolution: new developments in drug development for psychiatry
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 23, 2019 Category: Drugs & Pharmacology Authors: Linda S. Brady William Z. Potter Joshua A. Gordon Source Type: research

Estimating human ADME properties, pharmacokinetic parameters and likely clinical dose in drug discovery
Volume 14, Issue 12, December 2019, Page 1313-1327 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 20, 2019 Category: Drugs & Pharmacology Authors: Adam J. Lucas Joanne L. Sproston Patrick Barton Robert J. Riley Source Type: research

PROTACs – a game-changing technology
Volume 14, Issue 12, December 2019, Page 1255-1268 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 20, 2019 Category: Drugs & Pharmacology Authors: Markella Konstantinidou Jingyao Li Bidong Zhang Zefeng Wang Shabnam Shaabani Frans Ter Brake Khaled Essa Alexander D ömling Source Type: research

Estimating human ADME properties, pharmacokinetic parameters and likely clinical dose in drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 20, 2019 Category: Drugs & Pharmacology Authors: Adam J. Lucas Joanne L. Sproston Patrick Barton Robert J. Riley Source Type: research

PROTACs – a game-changing technology
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 20, 2019 Category: Drugs & Pharmacology Authors: Markella Konstantinidou Jingyao Li Bidong Zhang Zefeng Wang Shabnam Shaabani Frans Ter Brake Khaled Essa Alexander D ömling Source Type: research

Correction
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 18, 2019 Category: Drugs & Pharmacology Source Type: research

How plausible is an Alzheimer ’s disease vaccine?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 17, 2019 Category: Drugs & Pharmacology Authors: Ram ón Cacabelos Source Type: research

Fragment-based screening with natural products for novel anti-parasitic disease drug discovery
Volume 14, Issue 12, December 2019, Page 1283-1295 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Miaomiao Liu Ronald J. Quinn Source Type: research

Induced degradation of protein kinases by bifunctional small molecules: a next-generation strategy
Volume 14, Issue 12, December 2019, Page 1237-1253 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Jay C. Groppe Source Type: research

4D- quantitative structure –activity relationship modeling: making a comeback
Volume 14, Issue 12, December 2019, Page 1227-1235 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Denis Fourches Jeremy Ash Source Type: research

4D- quantitative structure –activity relationship modeling: making a comeback
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Denis Fourches Jeremy Ash Source Type: research

Induced degradation of protein kinases by bifunctional small molecules: a next-generation strategy
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Jay C. Groppe Source Type: research

Fragment-based screening with natural products for novel anti-parasitic disease drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 12, 2019 Category: Drugs & Pharmacology Authors: Miaomiao Liu Ronald J. Quinn Source Type: research

Targeting the receptor-based interactome of the dopamine D1 receptor: looking for heteromer-selective drugs
Volume 14, Issue 12, December 2019, Page 1297-1312 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 11, 2019 Category: Drugs & Pharmacology Authors: Ver ònica Casadó-Anguera Antoni Cort és Vicent Casad ó Estefan ía Moreno Source Type: research

Targeting the receptor-based interactome of the dopamine D1 receptor: looking for heteromer-selective drugs
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 11, 2019 Category: Drugs & Pharmacology Authors: Ver ònica Casadó-Anguera Antoni Cort és Vicent Casad ó Estefan ía Moreno Source Type: research

The current impact of water thermodynamics for small-molecule drug discovery
Volume 14, Issue 12, December 2019, Page 1221-1225 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 10, 2019 Category: Drugs & Pharmacology Authors: Stefan Geschwindner Johan Ulander Source Type: research

The current impact of water thermodynamics for small-molecule drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - September 10, 2019 Category: Drugs & Pharmacology Authors: Stefan Geschwindner Johan Ulander Source Type: research

Recent progress and challenges in drug development to fight hand, foot and mouth disease
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 31, 2019 Category: Drugs & Pharmacology Authors: Ze Qin Lim Qing Yong Ng Justin Wei Qing Ng Vikneswari Mahendran Sylvie Alonso Source Type: research

Advances in the structural annotation of human carbonic anhydrases and impact on future drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 22, 2019 Category: Drugs & Pharmacology Authors: Alessio Nocentini Claudiu T. Supuran Source Type: research

Dealing with frequent hitters in drug discovery: a multidisciplinary view on the issue of filtering compounds on biological screenings
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 16, 2019 Category: Drugs & Pharmacology Authors: Rafael Ferreira Dantas Tereza Cristina Santos Evangelista Bruno Junior Neves Mario Roberto Senger Carolina Horta Andrade Sabrina Baptista Ferreira Floriano Paes Silva-Junior Source Type: research

An overview of late-stage functionalization in today ’s drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 14, 2019 Category: Drugs & Pharmacology Authors: Michael Moir Jonathon J. Danon Tristan A. Reekie Michael Kassiou Source Type: research

Advances in preclinical approaches to Chagas disease drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 14, 2019 Category: Drugs & Pharmacology Authors: Fernando Villalta Girish Rachakonda Source Type: research

An overview of late-stage functionalization in today ’s drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 14, 2019 Category: Drugs & Pharmacology Authors: Michael Moir Jonathon J. Danon Tristan A. Reekie Michael Kassiou Source Type: research

Advances in preclinical approaches to Chagas disease drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 14, 2019 Category: Drugs & Pharmacology Authors: Fernando Villalta Girish Rachakonda Source Type: research

Preclinical discovery and development of fingolimod for the treatment of multiple sclerosis
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 7, 2019 Category: Drugs & Pharmacology Authors: Claudia Volpi Ciriana Orabona Antonio Macchiarulo Roberta Bianchi Paolo Puccetti Ursula Grohmann Source Type: research

What human blood-brain barrier models can tell us about BBB function and drug discovery?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 6, 2019 Category: Drugs & Pharmacology Authors: Lino Ferreira Source Type: research

Advances with weak affinity chromatography for fragment screening
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - August 5, 2019 Category: Drugs & Pharmacology Authors: Fotios Tsopelas Anna Tsantili-Kakoulidou Source Type: research

How can monoclonal antibodies be harnessed against neglected tropical diseases and other infectious diseases?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 31, 2019 Category: Drugs & Pharmacology Authors: Andreas H. Laustsen Source Type: research

Novel approaches to anti-obesity drug discovery with gut hormones over the past 10 years
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 29, 2019 Category: Drugs & Pharmacology Authors: Frances Rose Stephen Bloom Tricia Tan Source Type: research

Recent advances in computational design of potent aromatase inhibitors: open-eye on endocrine-resistant breast cancers
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 24, 2019 Category: Drugs & Pharmacology Authors: Angelo Spinello Ida Ritacco Alessandra Magistrato Source Type: research

Developments with bead-based screening for novel drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 23, 2019 Category: Drugs & Pharmacology Authors: Dehua Pei George Appiah Kubi Source Type: research

The human gut microbiome – a new and exciting avenue in cardiovascular drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 18, 2019 Category: Drugs & Pharmacology Authors: Yu Du Xingxing Li Chunyan Su Li Wang Jiandong Jiang Bin Hong Source Type: research

Design of α-helical antimicrobial peptides with a high selectivity index
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 17, 2019 Category: Drugs & Pharmacology Authors: Davor Jureti ć Juraj Simuni ć Source Type: research

Challenges to drug discovery for celiac disease and approaches to overcome them
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 17, 2019 Category: Drugs & Pharmacology Authors: Luis Vaquero David Bernardo Francisco Le ón Laura Rodr íguez-Martín Bego ña Alvarez-Cuenllas Santiago Vivas Source Type: research

Design of α-helical antimicrobial peptides with a high selectivity index
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 17, 2019 Category: Drugs & Pharmacology Authors: Davor Jureti ć Juraj Simuni ć Source Type: research

Challenges to drug discovery for celiac disease and approaches to overcome them
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 17, 2019 Category: Drugs & Pharmacology Authors: Luis Vaquero David Bernardo Francisco Le ón Laura Rodr íguez-Martín Bego ña Alvarez-Cuenllas Santiago Vivas Source Type: research

Transforming cancer drug discovery with Big Data and AI
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - July 9, 2019 Category: Drugs & Pharmacology Authors: Paul Workman Albert A. Antolin Bissan Al-Lazikani Source Type: research