Vutrisiran: a new drug in the treatment landscape of hereditary transthyretin amyloid polyneuropathy
Volume 19, Issue 4, April 2024, Page 393-402 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 28, 2024 Category: Drugs & Pharmacology Authors: Violaine Plant é-BordeneuveValentine Perraina Department of Neurology, Henri Mondor University Hospital, AP-HP, Créteil, Franceb Mondor Biomedical Research Institute – IMRB, INSERM, U955 Team 10 “Biology of the Neuromuscular System”, Créteil, Fra Source Type: research

Vutrisiran: a new drug in the treatment landscape of hereditary transthyretin amyloid polyneuropathy
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 28, 2024 Category: Drugs & Pharmacology Authors: Violaine Plant é-BordeneuveValentine Perraina Department of Neurology, Henri Mondor University Hospital, AP-HP, Créteil, Franceb Mondor Biomedical Research Institute – IMRB, INSERM, U955 Team 10 “Biology of the Neuromuscular System”, Créteil, Fra Source Type: research

Molecular glue degraders: exciting opportunities for novel drug discovery
Volume 19, Issue 4, April 2024, Page 433-449 . (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 24, 2024 Category: Drugs & Pharmacology Authors: Thomas LemaitreMarie CornuFlorian SchwalenMarc SinceCharline KiefferAnne Sophie Voisin-Chireta Normandie University, UNICAEN, CERMN, Caen, Franceb Department of Pharmacy, Caen University Hospital, Caen, France Source Type: research

Advances in structure-activity relationships of HDAC inhibitors as HIV latency-reversing agents
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 23, 2024 Category: Drugs & Pharmacology Authors: Samima KhatunSk. Abdul AminDebasmita ChoudhuryBoby ChowdhuryTarun JhaShovanlal Gayena Laboratory of Drug Design and Discovery, Department of Pharmaceutical Technology, Jadavpur University, Kolkata, Indiab Department of Pharmaceutical Technology, JIS Unive Source Type: research

Molecular glue degraders: exciting opportunities for novel drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 19, 2024 Category: Drugs & Pharmacology Authors: Thomas LemaitreMarie CornuFlorian SchwalenMarc SinceCharline KiefferAnne Sophie Voisin-Chireta Normandie University, UNICAEN, CERMN, Caen, Franceb Department of Pharmacy, Caen University Hospital, Caen, France Source Type: research

Have spirocyclic scaffolds been properly utilized in recent drug discovery efforts?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 16, 2024 Category: Drugs & Pharmacology Authors: Erica BenedettiLaurent MicouinLaboratoire de Chimie et Biochimie Pharmacologiques et Toxicologiques, Universit é Paris Cité, CNRS, Paris, France Source Type: research

What is the future of click chemistry in drug discovery and development?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - January 12, 2024 Category: Drugs & Pharmacology Authors: Ana C. AmorimAnthony J. Burkea Chemistry Department, Coimbra Chemistry Centre, Institute of Molecular Sciences, Coimbra, Portugalb Faculty of Pharmacy, University of Coimbra, Coimbra, Portugalc LAQV-REQUIMTE, Institute for Research and Advanced Studies, U Source Type: research

Designing drugs optimized for both blood –brain barrier permeation and intra-cerebral partition
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 25, 2023 Category: Drugs & Pharmacology Authors: Maria DichiaraGiuseppe CosentinoGiorgia GiordanoLorella PasquinucciAgostino MarrazzoGiuliana CostanzoEmanuele AmataDipartimento di Scienze del Farmaco e della Salute, Universit à degli Studi di Catania, Catania, Italy Source Type: research

Vascular organs-on-chip made with patient-derived endothelial cells: technologies to transform drug discovery and disease modeling
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 20, 2023 Category: Drugs & Pharmacology Authors: Chloe P WhitworthWilliam J Polachecka Curriculum in Genetics and Molecular Biology, University of North Carolina at Chapel Hill, Chapel Hill, NC, USAb Joint Department of Biomedical Engineering, University of North Carolina at Chapel Hill, Chapel Hill, NC Source Type: research

The SH-SY5Y cell line: a valuable tool for Parkinson ’s disease drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 19, 2023 Category: Drugs & Pharmacology Authors: Manisha PandeyVarnita KarmakarAnkit MajieMonika DwivediShadab MdBapi Goraina Department of Pharmaceutical Sciences, Central University of Haryana, Mahendergarh, Indiab Department of Pharmaceutical Sciences and Technology, Birla Institute of Technology, Me Source Type: research

Ultra-high-throughput mass spectrometry in drug discovery: fundamentals and recent advances
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 19, 2023 Category: Drugs & Pharmacology Authors: Jon D. WilliamsFan PuJames W. SawickiNathaniel L. ElsenAbbvie Discovery Research, North Chicago, IL, USA Source Type: research

Advances in ion channel high throughput screening: where are we in 2023?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 18, 2023 Category: Drugs & Pharmacology Authors: Mark L DallasDamian Bella Reading School of Pharmacy, University of Reading, Reading, UKb Sophion Biosciences, Copenhagen, Denmark Source Type: research

The problem of antimalarial resistance and its implications for drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 18, 2023 Category: Drugs & Pharmacology Authors: Thomas Martin Sch äferLais Pessanha de CarvalhoJuliana InoueAndrea KreidenweissJana Helda Institute of Tropical Medicine, University of Tübingen, Tübingen, Germanyb Centre de Recherches Médicales de Lambaréné, Lambaréné, Gabonc German Center for I Source Type: research

Current views on in vivo models for breast cancer research and related drug development
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 14, 2023 Category: Drugs & Pharmacology Authors: Tiago FerreiraTiago AzevedoJessica SilvaAna I. Faustino-RochaPaula A. Oliveiraa Centre for the Research and Technology of Agro-Environmental and Biological Sciences (CITAB), University of Tr ás-os-Montes and Alto Douro (UTAD), Vila Real, Portugalb Instit Source Type: research

Perspectives on the success of plasma lipidomics in cardiovascular drug discovery and future challenges
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - December 13, 2023 Category: Drugs & Pharmacology Authors: Timothy AbrahamsStephen J. NichollsFrom the Victorian Heart Institute, Monash University, Melbourne, Australia Source Type: research