How can we unlock the full potential of marine biological resources for novel drug discovery in an effective and ethical way?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 23, 2023 Category: Drugs & Pharmacology Authors: Hidayat HussainDepartment of Bioorganic Chemistry, Leibniz Institute of Plant Biochemistry, Halle (Saale), Germany Source Type: research

Advances in drug structure-activity-relationships for the development of selenium-based compounds against HIV
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 21, 2023 Category: Drugs & Pharmacology Authors: Dazhou ShiShujing XuDang DingKai TangYang ZhouXiangyi JiangShuo WangXinyong LiuPeng ZhanDepartment of Medicinal Chemistry, Key Laboratory of Chemical Biology, Ministry of Education, School of Pharmaceutical Sciences, Shandong University, Jinan, PR China Source Type: research

The vinyl sulfone motif as a structural unit for novel drug design and discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 18, 2023 Category: Drugs & Pharmacology Authors: You-Cai XiaoFen-Er Chena Key Laboratory of Drug-Targeting and Drug Delivery System of the Ministry of Education and Sichuan Research Center for Drug Precision Industrial Technology, West China School of Pharmacy, Sichuan University, Chengdu, Chinab Engine Source Type: research

Successfully navigating the valley of death: the importance of accelerators to support academic drug discovery and development
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 16, 2023 Category: Drugs & Pharmacology Authors: Maaike EvertsMark DrewTranslational Therapeutics Accelerator (TRxA), Critical Path Institute, Tucson, AZ, USA Source Type: research

Artificial intelligence pushes the boundaries of behavioral analysis in drug discovery: a revolution from the deep
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 10, 2023 Category: Drugs & Pharmacology Authors: Kurt Leroy HoffmanCentro de Investigaci ón en Reproducción Animal, Universidad Autónoma de Tlaxcala – CINVESTAV, Tlaxcala, Mexico Source Type: research

Recent applications of positron emission tomographic (PET) imaging in psychiatric drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 10, 2023 Category: Drugs & Pharmacology Authors: Luc Zimmera Lyon Neuroscience Research Center, Universit é Claude Bernard, Lyon, Franceb CERMEP, Hospices Civils de Lyon, Lyon, Francec Institut National des Sciences et Technologies Nucléaire, Saclay, France Source Type: research

Current strategic trends in drug discovery: the present as prologue
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 8, 2023 Category: Drugs & Pharmacology Authors: David R. JaneroDepartment of Pharmaceutical Sciences, School of Pharmacy and Pharmaceutical Sciences, and Health Sciences Entrepreneurs, Northeastern University, Boston, MA, USA Source Type: research

Benford ’s Law and distributions for better drug design
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 3, 2023 Category: Drugs & Pharmacology Authors: Alfonso T. Garc ía-SosaChair of Molecular Technology, Institute of Chemistry, University of Tartu, Tartu, Estonia Source Type: research

In vitro screening technologies for the discovery and development of novel drugs against Toxoplasma gondii
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 3, 2023 Category: Drugs & Pharmacology Authors: Joachim M üllerAndrew HemphillInstitute of Parasitology, Department of Infectious Diseases and Pathobiology, Vetsuisse Faculty, University of Bern, Bern, Switzerland Source Type: research

Evaluating physiochemical properties of FDA-approved orally administered drugs
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 3, 2023 Category: Drugs & Pharmacology Authors: Tanner C. ReeseAnvita DevineniTristan SmithIsmail LalamiJung-Mo AhnGanesh V. Raja Department of Urology, University of Texas Southwestern Medical Center, Dallas, USAb Department of Chemistry and Biochemistry, University of Texas at Dallas, Richardson, USA Source Type: research

γ-Secretase: once and future drug target for Alzheimer’s disease
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - November 2, 2023 Category: Drugs & Pharmacology Authors: Michael S. WolfeDepartment of Medicinal Chemistry, University of Kansas, Lawrence Source Type: research

Generative artificial intelligence empowers digital twins in drug discovery and clinical trials
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - October 27, 2023 Category: Drugs & Pharmacology Authors: Maria BordukovaNikita MakarovRaul Rodriguez-EstebanFabian SchmichMichael P. Mendena Data & Analytics, Pharmaceutical Research and Early Development, Roche Innovation Center Munich (RICM), Penzberg, Germanyb Institute of Computational Biology, Computation Source Type: research

Generative artificial intelligence empowers digital twins in drug discovery and clinical trials:
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - October 27, 2023 Category: Drugs & Pharmacology Authors: Maria BordukovaNikita MakarovRaul Rodriguez-EstebanFabian SchmichMichael P. Mendena Data & Analytics, Pharmaceutical Research and Early Development, Roche Innovation Center Munich (RICM), Penzberg, Germanyb Institute of Computational Biology, Computation Source Type: research

Advancements in the use of xenopus oocytes for modelling neurological disease for novel drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - October 18, 2023 Category: Drugs & Pharmacology Authors: Eoin C O ’ConnorKumiko KambaraDaniel Bertranda Roche Pharma Research and Early Development, Neuroscience & Rare Diseases, Roche Innovation Center Basel, Basel, Switzerlandb Development, HiQScreen S àrl, Geneva, Switzerland Source Type: research

Drugs targeting the particle for arrangement of quaternary structure (PAQosome) and protein complex assembly
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - October 16, 2023 Category: Drugs & Pharmacology Authors: Maxime PinardAsmae MoursliBenoit Coulombea Translational Proteomics Laboratory, Institut de Recherches Cliniques de Montr éal, Montréal, Québec, Canadab Department of Biochemistry and Molecular Medicine, Université de Montréal, Montréal, Québec, Ca Source Type: research