Zebrafish for modeling stroke and their applicability for drug discovery and development
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - May 23, 2022 Category: Drugs & Pharmacology Authors: Siobhan Crilly Emily McMahon Paul R. Kasher Source Type: research

What are the challenges with multi-targeted drug design for complex diseases?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - May 12, 2022 Category: Drugs & Pharmacology Authors: Agata Zi ęba Piotr St ępnicki Dariusz Matosiuk Agnieszka A. Kaczor Source Type: research

An overview of the preclinical discovery and development of trastuzumab deruxtecan: a novel gastric cancer therapeutic
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - April 15, 2022 Category: Drugs & Pharmacology Authors: James Kalmuk Dan Rinder Carl Heltzel Albert Craig Lockhart Source Type: research

Emerging three-dimensional neuronal culture assays for neurotherapeutics drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - April 5, 2022 Category: Drugs & Pharmacology Authors: Rahul S Rathore Senthil R Ayyannan Sanjeev K Mahto Source Type: research

Preclinical discovery and development of the casirivimab + imdevimab cocktail for the treatment of novel coronavirus infection: the rise and fall
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - April 1, 2022 Category: Drugs & Pharmacology Authors: Marco Tuccori Irma Convertino Sara Ferraro Emiliano Cappello Giulia Valdiserra Giulia de Luca Massimo Franchini Daniele Focosi Source Type: research

Advances in the use of 3D colorectal cancer models for novel drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 28, 2022 Category: Drugs & Pharmacology Authors: Ana Bai ão Sofia Dias Ana Francisca Soares Catarina Leite Pereira Carla Oliveira Bruno Sarmento Source Type: research

Recent in vivo advances of spirocyclic scaffolds for drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 25, 2022 Category: Drugs & Pharmacology Authors: Vasco F. Batista Diana C. G. A. Pinto Artur M. S. Silva Source Type: research

The design and discovery of topoisomerase I inhibitors as anticancer therapies
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 24, 2022 Category: Drugs & Pharmacology Authors: Endika Mart ín-Encinas Asier Selas Francisco Palacios Concepci ón Alonso Source Type: research

Perspectives on the design and discovery of α-ketoamide inhibitors for the treatment of novel coronavirus: where do we stand and where do we go?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 21, 2022 Category: Drugs & Pharmacology Authors: Alessio Nocentini Clemente Capasso Claudiu T. Supuran Source Type: research

Animal models of systemic lupus erythematosus and their applications in drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 15, 2022 Category: Drugs & Pharmacology Authors: Yue Xin Bo Zhang Junpeng Zhao Qianmei Liu Haoyuan Yin Qianjin Lu Source Type: research

Antimicrobial peptides: A plausible approach for COVID-19 treatment
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 10, 2022 Category: Drugs & Pharmacology Authors: Pooja Rani Bhupinder Kapoor Monica Gulati Atanas G. Atanasov Qushmua Alzahrani Reena Gupta Source Type: research

Natural products as novel scaffolds for the design of glycogen synthase kinase 3 β inhibitors
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 9, 2022 Category: Drugs & Pharmacology Authors: Serena Montanari Claudia Seidl Lara Davani Eleonora Gianquinto Eliska Emrichova Cristina Terenzi Vincenza Andrisano Angela De Simone Source Type: research

Targeting the cytoskeleton and extracellular matrix in cardiovascular disease drug discovery
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 8, 2022 Category: Drugs & Pharmacology Authors: Bohdan B. Khomtchouk Yoon Seo Lee Maha L. Khan Patrick Sun Deniel Mero Michael H. Davidson Source Type: research

What are the current challenges for machine learning in drug discovery and repurposing?
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 8, 2022 Category: Drugs & Pharmacology Authors: Tero Aittokallio Source Type: research

In silico drug discovery of melatonin receptor ligands with therapeutic potential
. (Source: Expert Opinion on Drug Discovery)
Source: Expert Opinion on Drug Discovery - March 8, 2022 Category: Drugs & Pharmacology Authors: Gian Marco Elisi Laura Scalvini Alessio Lodola Annalida Bedini Gilberto Spadoni Silvia Rivara Source Type: research