The search for brain-permeant NKCC1 inhibitors for the treatment of seizures: Pharmacokinetic-pharmacodynamic modelling of NKCC1 inhibition by azosemide, torasemide, and bumetanide in mouse brain

Publication date: Available online 2 December 2020Source: Epilepsy & BehaviorAuthor(s): Philip Hampel, Kerstin Römermann, Martina Gramer, Wolfgang Löscher
Source: Epilepsy and Behavior - Category: Neurology Source Type: research