[ASAP] Structure-Based Drug Discovery of < italic toggle="yes" > N < /italic > -(( < italic toggle="yes" > R < /italic > )-3-(7-Methyl-1 < italic toggle="yes" > H < /italic > -indazol-5-yl)-1-oxo-1-((( < italic toggle="yes" > S < /italic > )-1-oxo-3-(piperidin-4-yl)-1-(4-(pyridin-4-yl)piperazin-1-yl)propan-2-yl)amino)propan-2-yl)-2'-oxo-1',2'-dihydrospiro[piperidine-4,4'-pyrido[2,3- < italic toggle="yes" > d < /italic > ][1,3]oxazine]-1-carboxamide (HTL22562): A Calcitonin Gene-Related Peptide Receptor Antagonist for Acute Treatment of Migraine
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.0c01003
Source: Journal of Medicinal Chemistry - Category: Chemistry Authors: Sarah J. Bucknell* †, Mark A. Ator‡§, Alastair J. H. Brown†, Jason Brown†, Andrew D. Cansfield†, Julie E. Cansfield†, John A. Christopher†, Miles Congreve†, Gabriella Cseke†, Francesca Deflorian†, Christopher R. Jones†?, Jonathan S. Source Type: research