Palladium-catalyzed C-glycosylation and annulation of o-alkynylanilines with 1-iodoglycals: convenient access to 3-indolyl-C-glycosides

Org. Biomol. Chem., 2020, Accepted Manuscript DOI: 10.1039/D0OB01812K, CommunicationJianchao Liu, Xiao Xiao, Puren Han, Huiwen Zhou, Qi-Shuang Yin, Jian-Song Sun An efficient and practical approach for the synthesis of 3-indolyl-C- ∆1,2–glycosides through a palladium-catalyzed annulation/C-glycosylation sequence of o-alkynylanilines with 1-iodoglycals has been developed. This methodology has a wide scope of substrates... The content of this RSS Feed (c) The Royal Society of Chemistry

Source: RSC - Organic and Biomolecular Chemistry - October 19, 2020 Category: Molecular Biology Authors: Jianchao Liu Source Type: research