[ASAP] Discovery of ARD-2051 as a Potent and Orally Efficacious Proteolysis Targeting Chimera (PROTAC) Degrader of Androgen Receptor for the Treatment of Advanced Prostate Cancer

Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.3c00405

Source: Journal of Medicinal Chemistry - June 29, 2023 Category: Chemistry Authors: Xin Han, Lijie Zhao, Weiguo Xiang, Bukeyan Miao, Chong Qin □, Mi Wang, Tianfeng Xu, Donna McEachern, Jianfeng Lu, Yu Wang, Hoda Metwally, Chao-Yie Yang△, Paul D. Kirchhoff, Lu Wang, Aleksas Matvekas, John Takyi-Williams, Bo Wen, Duxin Sun, Mark Ator, Source Type: research