Toxic metabolites and metabolic soft spots of celastrol based on glutathione metabolic capture and high-resolution mass spectrometry
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 25, 2023 Category: Drugs & Pharmacology Authors: Xiaojuan JiangCaixia YuanRong DingDi LuXiaoyu PengZhihao DongChunyan ZhuYihua LinCaisheng WuQiang Xiea Fujian Provincial Key Laboratory of Innovative Drug Target Research and State Key Laboratory of Cell Stress Biology, School of Pharmaceutical Sciences, Source Type: research

Where developmental toxicity meets explainable artificial intelligence: state-of-the-art and perspectives
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 23, 2023 Category: Drugs & Pharmacology Authors: Maria Vittoria TogoFabrizio MastroloritoAngelica OrfinoElisabetta Anna GrapsAnna Rita TondoCosimo Damiano AltomareFulvio CiriacoDaniela TrisciuzziOrazio NicolottiNicola Amorosoa Department of Pharmacy - Pharmaceutical Sciences, Universit à degli Studi di Source Type: research

A pharmacokinetic evaluation of tenapanor for the treatment of irritable bowel syndrome with constipation: an update of the literature
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 18, 2023 Category: Drugs & Pharmacology Authors: Diego Curr òGianluca IaniroAntonio Gasbarrinia Pharmacology Section, Department of Health Care Surveillance and Bioethics, Università Cattolica del Sacro Cuore, Rome, Italyb Department of Translational Medicine and Surgery, Università Cattolica del Sac Source Type: research

Overcoming barriers to machine learning applications in toxicity prediction
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 13, 2023 Category: Drugs & Pharmacology Authors: Abdallah Abou HajalAhmad Z. Al Meslamania College of Pharmacy, Al Ain University, Abu Dhabi, United Arab Emiratesb AAU Health and Biomedical Research Center, Al Ain University, Abu Dhabi, United Arab Emirates Source Type: research

Pharmacokinetic evaluation of sofosbuvir/velpatasvir for the treatment of Chronic Hepatitis C in pediatrics aged 3 and older
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 7, 2023 Category: Drugs & Pharmacology Authors: Jessica TuanAdaora OkoliOnyema Ogbuagua Yale School of Medicine, Department of Internal Medicine, Section of Infectious Diseases, New Haven, CT, USAb Yale AIDS Program, 135 College St, New Haven, CT, USA Source Type: research

Evaluation of bioequivalence and safety analysis of capecitabine tablets and Xeloda ® under postprandial dosing conditions in Chinese patients with solid tumor
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 7, 2023 Category: Drugs & Pharmacology Authors: Hongtao LiRongfang ShanJiaxiang DingJialin ZhangBingyan LiuQin GeDongmei ChengLufeng LiChaoyang ZhangHe SuXiaoyue LiHuiru LiJingjing YeHui LiFengxian LiHuan ZhouQiang HuoYue Sua National Institute of Clinical Drug Trials, The First Affiliated Hospital of Source Type: research

CYP3A inhibitor itraconazole affect pharmacokinetic behavior of famitinib and its active metabolite: results of a single-center, single-arm, open-label and fixed sequence study
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - December 6, 2023 Category: Drugs & Pharmacology Authors: Yunzhe HuangYuanwei JiaXinyan ChenChangmao WangYaqin WangMinhui WangPing WuJie Shena Anhui provincial Center of Drug Clinical Evaluation, Yijishan Hospital of Wannan Medical College, Wuhu, Anhui, People ’s Republic of Chinab School of pharmacy, Wannan M Source Type: research

Drug-drug interactions between COVID-19 therapeutics and psychotropic medications
. (Source: Expert Opinion on Drug Metabolism and Toxicology)
Source: Expert Opinion on Drug Metabolism and Toxicology - November 30, 2023 Category: Drugs & Pharmacology Authors: Alessandro CuomoGiovanni Barill àGianluca SerafiniAndrea AgugliaAndrea AmerioMatteo CattolicoPietro CarmelliniAlessandro SpitiAndrea Fagiolinia Division of Psychiatry, Department of Molecular Medicine University of Siena School of Medicine Siena, Siena, Source Type: research