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Source: Molecular Pharmaceutics

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Total 100 results found since Jan 2013.

ASAP Silencing of Gasdermin D by siRNA-Loaded PEI-Chol Lipopolymers Potently Relieves Acute Gouty Arthritis through Inhibiting Pyroptosis
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.0c00229
Source: Molecular Pharmaceutics - July 6, 2020 Category: Drugs & Pharmacology Authors: Shu-Min Ye †‡#, Meng-Ze Zhou†#, Wen-Jiao Jiang†, Chun-Xiao Liu†‡, Zhan-Wei Zhou‡, Min-Jie Sun*‡, and Qing-Hua Hu*†‡ Source Type: research

ASAP Monoclonal Antibody 2C5-Modified Mixed Dendrimer Micelles for Tumor-Targeted Codelivery of Chemotherapeutics and siRNA
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.0c00075
Source: Molecular Pharmaceutics - April 10, 2020 Category: Drugs & Pharmacology Authors: Jiayi Pan †, Sara Aly Attia†, Md Abdus Subhan†‡, Nina Filipczak†§, Livia Palmerston Mendes†?, Xiang Li†#, Satya Siva Kishan Yalamarty†, and Vladimir P. Torchilin*†? Source Type: research

ASAP Polyarginine-Mediated siRNA Delivery: A Mechanistic Study of Intracellular Trafficking of PCL-R15/siRNA Nanoplexes
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.0c00120
Source: Molecular Pharmaceutics - March 30, 2020 Category: Drugs & Pharmacology Authors: Hai-Tao Zhang †‡§, Minzhi Yu‡, Yu-Jie Niu‡, Wei-Zhong Liu‡, Wen-Hao Pang‡, Jinsong Ding*†, and Jian-Cheng Wang*‡ Source Type: research

ASAP Compression of Vectors for Small Interfering RNAs Delivery: Toward Oral Administration of siRNA Lipoplexes in Tablet Forms
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.9b01190
Source: Molecular Pharmaceutics - March 16, 2020 Category: Drugs & Pharmacology Authors: Virginie Busignies †, Danielle Campiol Arruda‡§, Christine Charrueau§, Marcela Coelho Silva Ribeiro‡§, Anne-Marie Lachage`s§, Angelo Malachias?, Ste´phanie Finet?, Asad Ur Rehman§, Pascal Bigey§#, Pierre Tchoreloff†, and Virginie Escriou*§ Source Type: research

ASAP Improved Stability of siRNA-Loaded Lipid Nanoparticles Prepared with a PEG-Monoacyl Fatty Acid Facilitates Ligand-Mediated siRNA Delivery
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.0c00087
Source: Molecular Pharmaceutics - March 2, 2020 Category: Drugs & Pharmacology Authors: Yu Sakurai* †, Wataru Mizumura†, Kenichiro Ito‡, Kazuhiro Iwasaki§, Takayuki Katoh‡, Yuki Goto‡, Hiroaki Suga‡, and Hideyoshi Harashima*† Source Type: research

ASAP Construction of a Targeting Nanoparticle of 3',3?-Bis-Peptide-siRNA Conjugate/Mixed Lipid with Postinserted DSPE-PEG2000-cRGD
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.9b00800
Source: Molecular Pharmaceutics - November 6, 2019 Category: Drugs & Pharmacology Authors: Yanfen Zhang †‡§, Sixiu Li†§, Xinyang Zhou†§, Jing Sun†, Xinmeng Fan†, Zhu Guan†, Lihe Zhang†, and Zhenjun Yang*† Source Type: research

ASAP Effect of the Ratio of Betamethasone to TNF-a siRNA Coencapsulated in Solid Lipid Nanoparticles on the Acute Proinflammatory Activity of the Nanoparticles
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.9b00629
Source: Molecular Pharmaceutics - September 30, 2019 Category: Drugs & Pharmacology Authors: Hannah L. O ’Mary†, Mahmoud S. Hanafy†, Abdulaziz M. Aldayel†‡, Solange A. Valdes†, Riyad F. Alzhrani†, Stephanie Hufnagel†, John J. Koleng§, and Zhengrong Cui*† Source Type: research

ASAP A Multifunctional Lipid-Based Nanodevice for the Highly Specific Codelivery of Sorafenib and Midkine siRNA to Hepatic Cancer Cells
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.9b00738
Source: Molecular Pharmaceutics - August 23, 2019 Category: Drugs & Pharmacology Authors: Mahmoud A. Younis †$, Ikramy A. Khalil*†$, Mahmoud M. Abd Elwakil†, and Hideyoshi Harashima*† Source Type: research

ASAP Self-Assembled Cationic ß-Cyclodextrin Nanostructures for siRNA Delivery
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.8b01307
Source: Molecular Pharmaceutics - February 19, 2019 Category: Drugs & Pharmacology Authors: Raghvendra Pratap Singh, Tania Hidalgo, Pierre-Andre Cazade, Raphael Darcy, Michael F. Cronin, Irina Dorin, Caitr íona M. O’Driscoll, Damien Thompson Source Type: research

ASAP Synergistic Targeting HER2 and EGFR with Bivalent Aptamer-siRNA Chimera Efficiently Inhibits HER2-Positive Tumor Growth
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.8b00388
Source: Molecular Pharmaceutics - October 1, 2018 Category: Drugs & Pharmacology Authors: Lu Xue, Nita J. Maihle, Xiaolin Yu, Shou-Ching Tang, Hong Yan Liu Source Type: research

ASAP A Glutamine-Rich Carrier Efficiently Delivers Anti-CD47 siRNA Driven by a “Glutamine Trap” To Inhibit Lung Cancer Cell Growth
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.8b00076
Source: Molecular Pharmaceutics - July 6, 2018 Category: Drugs & Pharmacology Authors: Jiamin Wu, Zhi Li, Zeping Yang, Ling Guo, Ye Zhang, Huihui Deng, Cuifeng Wang, Min Feng Source Type: research

ASAP Reducing the Cytotoxicity of Lipid Nanoparticles Associated with a Fusogenic Cationic Lipid in a Natural Killer Cell Line by Introducing a Polycation-Based siRNA Core
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.7b01166
Source: Molecular Pharmaceutics - April 30, 2018 Category: Drugs & Pharmacology Authors: Takashi Nakamura, Koharu Yamada, Yuki Fujiwara, Yusuke Sato, Hideyoshi Harashima Source Type: research

Systemic Administration of siRNA with Anti-HB-EGF Antibody-Modified Lipid Nanoparticles for the Treatment of Triple-Negative Breast Cancer
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.7b01055
Source: Molecular Pharmaceutics - March 12, 2018 Category: Drugs & Pharmacology Authors: Ayaka Okamoto, Tomohiro Asai, Yusuke Hirai, Kosuke Shimizu, Hiroyuki Koide, Tetsuo Minamino and Naoto Oku Source Type: research

ASAP Systemic Administration of siRNA with Anti-HB-EGF Antibody-Modified Lipid Nanoparticles for the Treatment of Triple-Negative Breast Cancer
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.7b01055
Source: Molecular Pharmaceutics - March 12, 2018 Category: Drugs & Pharmacology Authors: Ayaka Okamoto, Tomohiro Asai, Yusuke Hirai, Kosuke Shimizu, Hiroyuki Koide, Tetsuo Minamino, Naoto Oku Source Type: research

High-Content Surface and Total Expression siRNA Kinase Library Screen with VX-809 Treatment Reveals Kinase Targets that Enhance F508del-CFTR Rescue
Molecular PharmaceuticsDOI: 10.1021/acs.molpharmaceut.7b00928
Source: Molecular Pharmaceutics - February 9, 2018 Category: Drugs & Pharmacology Authors: Lydia A. Perkins, Gregory W. Fisher, Matharishwan Naganbabu, Brigitte F. Schmidt, Frederick Mun and Marcel P. Bruchez Source Type: research