The role of caveolin-1 in the biofate and efficacy of anti-tumor drugs and their nano-drug delivery systems
Publication date: Available online 28 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Canyu Yang, Bing He, Wenbing Dai, Hua Zhang, Ying Zheng, Xueqing Wang, Qiang Zhang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 29, 2020 Category: Cancer & Oncology Source Type: research

Targeting BMI-1-mediated epithelial–mesenchymal transition to inhibit colorectal cancer liver metastasis
Publication date: Available online 28 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Zhiyao Xu, Zhuha Zhou, Jing Zhang, Feichao Xuan, Mengjing Fan, Difan Zhou, Zhengyu Liuyang, Ximei Ma, Yiyang Hong, Yihong Wang, Sherven Sharma, Qinghua Dong, Guanyu Wang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 29, 2020 Category: Cancer & Oncology Source Type: research

Recent advances in nanomedicines for the treatment of ischemic stroke
Publication date: Available online 28 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Chao Li, Chen Jiang, Tao Sun (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 29, 2020 Category: Cancer & Oncology Source Type: research

Targeting redox-altered plasticity to reactivate synaptic function: A novel therapeutic strategy for cognitive disorder
Publication date: Available online 24 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Pei Wang, Fang Wang, Lan Ni, Pengfei Wu, Jianguo Chen (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 25, 2020 Category: Cancer & Oncology Source Type: research

TPGS/hyaluronic acid dual-functionalized PLGA nanoparticles delivered through dissolving microneedles for markedly improved chemo-photothermal combined therapy of superficial tumor
Publication date: Available online 24 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Tingting Peng, Yao Huang, Xiaoqian Feng, Chune Zhu, Shi Yin, Xinyi Wang, Xuequn Bai, Xin Pan, Chuanbin Wu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 25, 2020 Category: Cancer & Oncology Source Type: research

Molecularly engineered truncated tissue factor with therapeutic aptamers for tumor-targeted delivery and vascular infarction
Publication date: Available online 24 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Bozhao Li, Jingyan Wei, Chunzhi Di, Zefang Lu, Feilong Qi, Yinlong Zhang, Wei Sun Leong, Lele Li, Guangjun Nie, Suping Li (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 25, 2020 Category: Cancer & Oncology Source Type: research

The disruption of protein−protein interactions with co-chaperones and client substrates as a strategy towards Hsp90 inhibition
Publication date: Available online 24 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Michael A. Serwetnyk, Brian S.J. Blagg (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 25, 2020 Category: Cancer & Oncology Source Type: research

Enzyme-instructed hybrid nanogel/nanofiber oligopeptide hydrogel for localized protein delivery
Publication date: Available online 21 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Tianyue Jiang, Yudi Ma, Xiao Xu, Qingchun Ji, Mingxing Feng, Cheng Cheng, Yang Feng, Bingfang He, Ran Mo (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 22, 2020 Category: Cancer & Oncology Source Type: research

Design, synthesis, and biological evaluation of Bcr-Abl PROTACs to overcome T315I mutation
Publication date: Available online 20 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Liang Jiang, Yuting Wang, Qian Li, Zhengchao Tu, Sihua Zhu, Sanfang Tu, Zhang Zhang, Ke Ding, Xiaoyun Lu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 21, 2020 Category: Cancer & Oncology Source Type: research

Uptake and trafficking of different sized PLGA nanoparticles by dendritic cells in imiquimod-induced psoriasis-like mice model
Publication date: Available online 20 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Zibei Lin, Long Xi, Shaokui Chen, Jinsong Tao, Yan Wang, Xin Chen, Ping Li, Zhenping Wang, Ying Zheng (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 21, 2020 Category: Cancer & Oncology Source Type: research

Facile synthesis of insulin fusion derivatives through sortase A ligation
Publication date: Available online 21 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Maria M. Disotuar, Jake A. Smith, Jinze Li, Steve Alam, Nai-Pin Lin, Danny Hung-Chieh Chou (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 21, 2020 Category: Cancer & Oncology Source Type: research

Abrogation of USP7 is an alternative strategy to downregulate PD-L1 and sensitize gastric cancer cells to T cells killing
Publication date: Available online 16 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Zhiru Wang, Wenting Kang, Ouwen Li, Fengyu Qi, Junwei Wang, Yinghua You, Pengxing He, Zhenhe Suo, Yichao Zheng, Hongmin Liu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 18, 2020 Category: Cancer & Oncology Source Type: research

Discovery of 4-arylthiophene-3-carboxylic acid as inhibitor of ANO1 and its effect as analgesic agent
Publication date: Available online 17 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Yuxi Wang, Jian Gao, Song Zhao, Yan Song, Han Huang, Guiwang Zhu, Peili Jiao, Xiangqing Xu, Guisen Zhang, Kewei Wang, Liangren Zhang, Zhenming Liu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 18, 2020 Category: Cancer & Oncology Source Type: research

Neutralizing antibodies for the treatment of COVID-19
Publication date: Available online 16 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Zeqi Zhou, Xiangbin Wang, Yankai Fu, Xiqing Zhang, Changxiao Liu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 16, 2020 Category: Cancer & Oncology Source Type: research

S-allylmercaptocysteine improves alcoholic liver disease partly through a direct modulation of insulin receptor signaling
Publication date: Available online 13 November 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Pingping Luo, Ming Zheng, Rui Zhang, Hong Zhang, Yingxia Liu, Wei Li, Xiaoming Sun, Qian Yu, George L. Tipoe, Jia Xiao (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 15, 2020 Category: Cancer & Oncology Source Type: research