Profibrotic mechanisms of DPP8 and DPP9 highly expressed in the proximal renal tubule epithelial cells
Publication date: Available online 29 April 2021Source: Pharmacological ResearchAuthor(s): Yuzhan Zhang, Ke Li, Yan Li, Weihao Zhao, Li Wang, Zhao Chen, Xiaotao Ma, Tian Yao, Jinhua Wang, Wei Dong, Xiancheng Li, Xuefei Tian, Rongguo Fu (Source: Pharmacological Research)
Source: Pharmacological Research - April 29, 2021 Category: Drugs & Pharmacology Source Type: research

Novel STAT3 Small-Molecule Inhibitors Identified by Structure-Based Virtual Ligand Screening Incorporating SH2 Domain Flexibility
Publication date: Available online 29 April 2021Source: Pharmacological ResearchAuthor(s): Ren Kong, Uddalak Bharadwaj, T Kris Eckols, Mikhail Kolosov, Haoyi Wu, Francisco J. Santa Cruz-Pavlovich, Alison Shaw, Oluwatomilona I. Ifelayo, Hong Zhao, Moses M. Kasembeli, Stephen T.C. Wong, David J Tweardy (Source: Pharmacological Research)
Source: Pharmacological Research - April 29, 2021 Category: Drugs & Pharmacology Source Type: research

New Application of an Old Drug Proparacaine in Treating Epilepsy via Liposomal Hydrogel Formulation
Publication date: Available online 29 April 2021Source: Pharmacological ResearchAuthor(s): Abdoh Taleb, Ya-Ping Zhou, Ling-Tong Meng, Ming-Yi Zhu, Qiao Zhang, Muhammad Naveed, Lian-Di Li, Qi-Gang Zhou, Fan Meng, Feng Han (Source: Pharmacological Research)
Source: Pharmacological Research - April 29, 2021 Category: Drugs & Pharmacology Source Type: research

BACH1 is transcriptionally inhibited by TET1 in hepatocellular carcinoma in a microRNA-34a-dependent manner to regulate autophagy and inflammation
Publication date: July 2021Source: Pharmacological Research, Volume 169Author(s): Xuehu Sun, Hongmei Zhu, Rongge Cao, Jianlin Zhang, Xingyu Wang (Source: Pharmacological Research)
Source: Pharmacological Research - April 29, 2021 Category: Drugs & Pharmacology Source Type: research

Medioresinol as a novel PGC-1α activator prevents pyroptosis of endothelial cells in ischemic stroke through PPARα-GOT1 axis
Publication date: Available online 27 April 2021Source: Pharmacological ResearchAuthor(s): Yunjie Wang, Xin Guan, Cheng-Long Gao, Wenchen Ruan, Shunyi Zhao, Guoyin Kai, Fei Li, Tao Pang (Source: Pharmacological Research)
Source: Pharmacological Research - April 28, 2021 Category: Drugs & Pharmacology Source Type: research

New Insights into the Hippo/YAP Pathway in Idiopathic Pulmonary Fibrosis
Publication date: Available online 27 April 2021Source: Pharmacological ResearchAuthor(s): Mingyao Sun, Yangyang Sun, Ziru Feng, Xinliang Kang, Weijie Yang, Yongan Wang, Yuan Luo (Source: Pharmacological Research)
Source: Pharmacological Research - April 28, 2021 Category: Drugs & Pharmacology Source Type: research

Didymin switches M1-like toward M2-like macrophage to ameliorate ulcerative colitis via fatty acid oxidation
Publication date: Available online 27 April 2021Source: Pharmacological ResearchAuthor(s): Qi Lv, Yao Xing, Yijun Liu, Qingzhu Chen, Jingyi Xu, Lihong Hu, Yinan Zhang (Source: Pharmacological Research)
Source: Pharmacological Research - April 28, 2021 Category: Drugs & Pharmacology Source Type: research

Compromised right ventricular contractility in an ovine model of heart transplantation following 24 hours donor brain stem death
Publication date: Available online 24 April 2021Source: Pharmacological ResearchAuthor(s): Matthew A Wells, Louise E See Hoe, Peter Molenaar, Sanne Pedersen, Nchafatso G Obonyo, Charles I McDonald, Weilan Mo, Mahè Bouquet, Kieran Hyslop, Margaret R Passmore, Nicole Bartnikowski, Jacky Y Suen, Jason N Peart, David C McGiffin, John F Fraser, on behalf of the Dead Heart Project (Source: Pharmacological Research)
Source: Pharmacological Research - April 25, 2021 Category: Drugs & Pharmacology Source Type: research

Editorial Board
Publication date: May 2021Source: Pharmacological Research, Volume 167Author(s): (Source: Pharmacological Research)
Source: Pharmacological Research - April 25, 2021 Category: Drugs & Pharmacology Source Type: research

Corrigendum to “Cannabidiol inhibits febrile seizure by modulating AMPA receptor kinetics through its interaction with the N-terminal domain of GluA1/GluA2” [Pharmacol. Res. 161 (2020) 105128 1-14]
Publication date: Available online 21 April 2021Source: Pharmacological ResearchAuthor(s): Yongzhou Yu, Zuxiao Yang, Baohua Jin, Xia Qin, Xiaoque Zhu, Jiahui Sun, Lifang Huo, Ri Wang, Yongyun Shi, Zhanfeng Jia, Yun Stone Shi, Shifeng Chu, Dezhi Kong, Wei Zhang (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research

Estrogen profile- and pharmacogenetics-based lamotrigine dosing regimen optimization: recommendations for pregnant women with epilepsy
Publication date: Available online 20 April 2021Source: Pharmacological ResearchAuthor(s): Ming-Lu Wang, Yu-Ying Tao, Xiao-Yu Sun, Yang Guo, Zhan-You Wang, Yun-Feng Cao, Limei Zhao (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research

Microvesicles – promising tiny players’ of cancer stem cells targeted liver cancer treatments: the interesting interactions and therapeutic aspects
Publication date: Available online 20 April 2021Source: Pharmacological ResearchAuthor(s): Cong He, Doulathunnisa Jaffar Ali, Smilin Bell Aseervatham G, Bo Sun, Zhongdang Xiao (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research

Liver organoid as a 3D in vitro model for drug validation and toxicity assessment
Publication date: Available online 20 April 2021Source: Pharmacological ResearchAuthor(s): Anastasia Brooks, Xiaowen Liang, Yonglong Zhang, Chun-Xia Zhao, Michael S. Roberts, Haolu Wang, Lei Zhang, Darrell H.G. Crawford (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research

Borneol in cardio-cerebrovascular diseases: pharmacological actions, mechanisms, and therapeutics
Publication date: Available online 21 April 2021Source: Pharmacological ResearchAuthor(s): Songyu Liu, Yu Long, Shuang Yu, Dingkun Zhang, Qiyue Yang, Zhimin Ci, Mingquan Cui, Yulu Zhang, Jinyan Wan, Dan Li, Ai Shi, Nan Li, Ming Yang, Junzhi Lin (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research

Mimicking bone microenvironment: 2D and 3D in vitro models of human osteoblasts
Publication date: Available online 21 April 2021Source: Pharmacological ResearchAuthor(s): I. Yuste, F.C. Luciano, E. González-Burgos, A. Lalatsa, D.R. Serrano (Source: Pharmacological Research)
Source: Pharmacological Research - April 22, 2021 Category: Drugs & Pharmacology Source Type: research