Co-spray dried hydrophobic drug formulations with crystalline lactose for inhalation aerosol delivery
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Wei-Ren Ke, Philip Chi Lip Kwok, Dipesh Khanal, Rachel Yoon Kyung Chang, Hak-Kim Chan (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Recent advances in mechanical force-assisted transdermal delivery of macromolecular drugs
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Ruxuan Wang, Qiong Bian, Yihua Xu, Donghang Xu, Jianqing Gao (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Determination of a quantitative relationship between material properties, process settings and screw feeding behavior via multivariate data-analysis
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): B.Bekaert, L. Penne, W. Grymonpré, B. Van Snick, J. Dhondt, J. Boeckx, J. Vogeleer, T. De Beer, C. Vervaet, V. Vanhoorne (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Soft Sensor for Real-Time Estimation of Tablet Potency in Continuous Direct Compression Manufacturing Operation
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Reza Kamyar, David Lauri Pla, Anas Husain, Giuseppe Cogoni, Zilong Wang (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Permeability-enhancing effects of three laurate-disaccharide monoesters across isolated rat intestinal mucosae
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Fiona McCartney, Diego R. Perinelli, Mattia Tiboni, Robert Cavanagh, Simone Lucarini, Giovanni Filippo Palmieri, Luca Casettari, David J. Brayden (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Characterisation and fundamental insight into the formation of new solid state, multicomponent systems of propranolol
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Klaudia Bialek, Zaneta Wojnarowska, Brendan Twamley, Lidia Tajber (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Oral administration of tipranavir with long-chain triglyceride results in moderate intestinal lymph targeting but no efficient delivery to HIV-1 reservoir in mesenteric lymph nodes
Publication date: Available online 21 April 2021Source: International Journal of PharmaceuticsAuthor(s): Yenju Chu, Chaolong Qin, Wanshan Feng, Charles Sheriston, Yu Jane Khor, Concepción Medrano-Padial, Birgit E. Watson, Teddy Chan, Binhua Ling, Michael J. Stocks, Peter M. Fischer, Pavel Gershkovich (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Controlling the release rate of topotecan from PLGA spheres and increasing its cytotoxicity towards glioblastoma cells by co-loading with calcium chloride
Publication date: Available online 21 April 2021Source: International Journal of PharmaceuticsAuthor(s): Racheli Sharon Gabbay, Abraham Rubinstein (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Thermosensitive and mucoadhesive in situ ocular gel for effective local delivery and antifungal activity of itraconazole nanocrystal in the treatment of fungal keratitis
Publication date: Available online 21 April 2021Source: International Journal of PharmaceuticsAuthor(s): Andi Dian Permana, Rifka Nurul Utami, Patricia Layadi, Achmad Himawan, Nana Juniarti, Qonita Kurnia Anjani, Emilia Utomo, Sandra Aulia Mardikasari, Andi Arjuna, Ryan F. Donnelly (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 21, 2021 Category: Drugs & Pharmacology Source Type: research

Protective effect of melatonin entrapped PLGA nanoparticles on radiation-induced lung injury through the the miR-21/TGF-β1/Smad3 pathway
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Shuang Wang, Juan Li, Yingjuan He, Yonghong Ran, Binghui Lu, Jining Gao, Chang Shu, Jie Li, Yazhen Zhao, Xin Zhang, Yuhui Hao (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research

The in vitro and in vivo study of novel formulation of Andrographolide PLGA nanoparticle embedded into gelatin-based hydrogel to prolong delivery and extend residence time in joint
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Thitianan Kulsirirat, Korbtham Sathirakul, Noriyasu Kamei, Mariko Takeda-Morishita (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research

Sounding Out Stability of Enteric Coated Dosage Forms using Broadband Acoustic Resonance Dissolution Spectroscopy (BARDS)
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Niamh O'Mahoney, Anas Alfarsi, Haley O'Sullivan, Seán McSweeney, Abina Crean, Dara Fitzpatrick (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research

Micelle-contained and PEGylated Hybrid Liposomes of Combined Gemcitabine and Cisplatin Delivery for enhancing antitumor activity
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Zixu Liu, Wei Chu, Qianhe Sun, Linxuan Zhao, Xinyi Tan, Yu Zhang, Tian Yin, Haibing He, Jingxin Gou, Xing Tang (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research

A straw for paediatrics: How to administer highly dosed, bitter tasting paracetamol granules
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Tilen Simšič, Boris Nolimal, Jasmina Minova, Ana Baumgartner, Odon Planinšek (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research

Paeonol-Loaded PLGA Nanoparticles as an Oral Drug Delivery System: Design, Optimization and Evaluation
Publication date: Available online 20 April 2021Source: International Journal of PharmaceuticsAuthor(s): Fangyuan Wang, Qianqian Shan, Xiangwei Chang, Zhenbao Li, Shuangying Gui (Source: International Journal of Pharmaceutics)
Source: International Journal of Pharmaceutics - April 20, 2021 Category: Drugs & Pharmacology Source Type: research