A multifunctional cross-validation high-throughput screening protocol enabling the discovery of new SHP2 inhibitors
Publication date: Available online 31 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Yihui Song, Min Zhao, Yahong Wu, Bin Yu, Hong-Min Liu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - November 1, 2020 Category: Cancer & Oncology Source Type: research

Hedgehog signaling in gastrointestinal carcinogenesis and the gastrointestinal tumor microenvironment
Publication date: Available online 29 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Jinghui Zhang, Jiajun Fan, Xian Zeng, Mingming Nie, Jingyun Luan, Yichen Wang, Dianwen Ju, Kai Yin (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 30, 2020 Category: Cancer & Oncology Source Type: research

Natural compounds modulate the autophagy with potential implication of stroke
Publication date: Available online 29 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Anil Ahsan, Mengru Liu, Yanrong Zheng, Wenping Yan, Lin Pan, Yue Li, Shijia Ma, Xingxian Zhang, Ming Cao, Zhanxun Wu, Weiwei Hu, Zhong Chen, Xiangnan Zhang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 30, 2020 Category: Cancer & Oncology Source Type: research

Impact of particle size and pH on protein corona formation of solid lipid nanoparticles: a proof-of-concept study
Publication date: Available online 29 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Wenhao Wang, Zhengwei Huang, Yanbei Li, Wenhua Wang, Jiayu Shi, Fangqin Fu, Ying Huang, Xin Pan, Chuanbin Wu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 30, 2020 Category: Cancer & Oncology Source Type: research

Author correction to ‘Cardamonin from a medicinal herb protects against LPS-induced septic shock by suppressing NLRP3 inflammasome’ [Acta Pharmaceutica Sinica B 9 (2019) 734–744]
Publication date: Available online 24 September 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Zhilei Wang, Guang Xu, Yuan Gao, Xiaoyan Zhan, Nan Qin, Shubin Fu, Ruisheng Li, Ming Niu, Jiabo Wang, Youping Liu, Xiaohe Xiao, Zhaofang Bai (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 23, 2020 Category: Cancer & Oncology Source Type: research

Escape from abluminal LRP1-mediated clearance for boosted nanoparticle brain delivery and brain metastasis treatment
Publication date: Available online 21 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Naveed Ullah Khan, Jiang Ni, Xiufeng Ju, Tongtong Miao, Haiyan Chen, Liang Han (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 21, 2020 Category: Cancer & Oncology Source Type: research

Reversible small-molecule polymerizable phosphatidylcholine: novel disulfide crosslinked micelles for redox-dependent drug delivery
Publication date: Available online 20 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Longbing Ling, Muhammad Ismail, Xinsong Li (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 20, 2020 Category: Cancer & Oncology Source Type: research

An injectable micelle-hydrogel hybrid for localized and prolonged drug delivery in the management of renal fibrosis
Publication date: Available online 18 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Xianyan Qin, Yingying Xu, Xu Zhou, Tao Gong, Zhi-Rong Zhang, Yao Fu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 20, 2020 Category: Cancer & Oncology Source Type: research

Nature’s marvels endowed in gaseous molecules I: carbon monoxide and its physiological and therapeutic roles
Publication date: Available online 16 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Xiaoxiao Yang, Wen Lu, Christopher P. Hopper, Bowen Ke, Binghe Wang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 17, 2020 Category: Cancer & Oncology Source Type: research

Discovery of a potent and dual-selective bisubstrate inhibitor for protein arginine methyltransferase 4/5
Publication date: Available online 16 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Ayad A. Al-Hamashi, Dongxing Chen, Youchao Deng, Guangping Dong, Rong Huang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 17, 2020 Category: Cancer & Oncology Source Type: research

GSH-responsive SN38 dimer-loaded shape-transformable nanoparticles with iRGD for enhancing chemo-photodynamic therapy
Publication date: Available online 15 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Congcong Lin, Fan Tong, Rui Liu, Rou Xie, Ting Lei, Yuxiu Chen, Zhihang Yang, Huile Gao, Xiangrong Yu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 17, 2020 Category: Cancer & Oncology Source Type: research

The phytochemical, biological, and medicinal attributes of phytoecdysteroids: an updated review
Publication date: Available online 16 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Niranjan Das, Siddhartha Kumar Mishra, Anusha Bishayee, Eunüs S. Ali, Anupam Bishayee (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 17, 2020 Category: Cancer & Oncology Source Type: research

Energy metabolism disorders and potential therapeutic drugs in heart failure
Publication date: Available online 14 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Yanan He, Wei Huang, Chen Zhang, Lumeng Chen, Runchun Xu, Nan Li, Fang Wang, Li Han, Ming Yang, Dingkun Zhang (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 15, 2020 Category: Cancer & Oncology Source Type: research

Design, synthesis, molecular modeling, and biological evaluation of acrylamide derivatives as potent inhibitors of human dihydroorotate dehydrogenase for the treatment of rheumatoid arthritis
Publication date: Available online 15 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Fanxun Zeng, Shiliang Li, Guantian Yang, Yating Luo, Tiantian Qi, Yingfan Liang, Tingyuan Yang, Letian Zhang, Rui Wang, Lili Zhu, Honglin Li, Xiaoyong Xu (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 15, 2020 Category: Cancer & Oncology Source Type: research

Angiotensin-converting enzyme 2 (ACE2): SARS-CoV-2 receptor and RAS modulator
Publication date: Available online 13 October 2020Source: Acta Pharmaceutica Sinica BAuthor(s): Jingwei Bian, Zijian Li (Source: Acta Pharmaceutica Sinica B)
Source: Acta Pharmaceutica Sinica B - October 15, 2020 Category: Cancer & Oncology Source Type: research