[ASAP] A Fluorescence Polarization Assay for Macrodomains Facilitates the Identification of Potent Inhibitors of the SARS-CoV ‑2 Macrodomain
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00092 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - May 1, 2023 Category: Chemistry Authors: Ananya Anmangandla, Sadhan Jana, Kewen Peng, Shamar D. Wallace, Saket R. Bagde, Bryon S. Drown, Jiashu Xu, Paul J. Hergenrother, J. Christopher Fromme, and Hening Lin Source Type: research

[ASAP] Bioactive Natural Product Discovery via Deuterium Adduct Bioactivity Screening
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00083 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - May 1, 2023 Category: Chemistry Authors: Nicholas A. Zill, Yongle Du, Samantha Marinkovich, Di Gu, Jeremy Seidel, and Wenjun Zhang Source Type: research

[ASAP] A Versatile Strategy to Manipulate and Probe Native Carbonic Anhydrases < italic toggle="yes" > In Cellulo < /italic > Utilizing Two-Step Ligand-Directed Functionalization
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00102 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - May 1, 2023 Category: Chemistry Authors: Wai-Seng Io and Tsung-Shing Andrew Wang Source Type: research

[ASAP] Discrimination of GLUTs by Fructose Isomers Enables Simultaneous Screening of GLUT5 and GLUT2 Activity in Live Cells
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00682 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 28, 2023 Category: Chemistry Authors: Nazar Gora, Lukasz J. Weselinski, Vagarshak V. Begoyan, Andrew Cooper, Jun-yong Choe, and Marina Tanasova Source Type: research

[ASAP] Chemoproteomics Reveals the Pan-HER Kinase Inhibitor Neratinib To Target an < italic toggle="yes" > Arabidopsis < /italic > Epoxide Hydrolase Related to Phytohormone Signaling
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00322 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 28, 2023 Category: Chemistry Authors: Sabrina Ninck, Vivek Halder, Jan H. Krahn, Daniela Beisser, Sarah Resch, Isobel Dodds, Rene ́ Scholtysik, Jenny Bormann, Leonard Sewald, Mainak D. Gupta, Geronimo Heilmann & , Deepak D. Bhandari, Kyoko Morimoto, Pierre Buscaill, Bettina Hause, Renier A. Source Type: research

[ASAP] Unexploited Performance of NLS in the dCas9-VPR-Mediated Transcriptional Activation
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00195 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 27, 2023 Category: Chemistry Authors: Junxiang Zhou, Miao He, Xue Yin, Yue Yu, Dongbao Yao, and Haojun Liang Source Type: research

[ASAP] SARS-CoV ‑2 Spike N‑Terminal Domain Engages 9‑ < italic toggle="yes" > O < /italic > ‑Acetylated α2–8-Linked Sialic Acids
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00066 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 27, 2023 Category: Chemistry Authors: Ilhan Tomris, Luca Unione, Linh Nguyen, Pouya Zaree, Kim M. Bouwman, Lin Liu, Zeshi Li, Jelle A. Fok, Mari ́a Ríos Carrasco, Roosmarijn van der Woude, Anne L. M. Kimpel, Mirte W. Linthorst, Sinan E. Kilavuzoglu, Enrico C. J. M. Verpalen, Tom G. Caniels Source Type: research

[ASAP] Palmitoylation-Dependent Small-Molecule Fluorescent Probes for Live-Cell Golgi Imaging
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00046 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 25, 2023 Category: Chemistry Authors: Shunsuke Sawada, Masaru Yoshikawa, Keita Tsutsui, Tomoki Miyazaki, Keiko Kano, Emi Mishiro-Sato, and Shinya Tsukiji Source Type: research

[ASAP] Discovery of Benzodiazepine-Based Inhibitors of the E2 Enzyme UBCH10 from a Cell-Based p21 Degradation Screen
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00909 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 25, 2023 Category: Chemistry Authors: Benoit Pelletier, Ste ́phanie Duhamel, Guillaume Tambutet, Scott Jarvis, Patrick Cléroux, Maud David, Pierre-Luc Tanguay, Laure Voisin, Clint James, Rico Lavoie, Yves Gareau, Joël Flynn-Robitaille, Thierry Lorca, Réjean Ruel, Anne Marinier, and Syl Source Type: research

[ASAP] Targeting Riboswitches with Beta-Axial-Substituted Cobalamins
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00939 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 24, 2023 Category: Chemistry Authors: Shelby R. Lennon, Aleksandra J. Wierzba, Shea H. Siwik, Dorota Gryko, Amy E. Palmer, and Robert T. Batey Source Type: research

[ASAP] Efficient Ligand Discovery Using Sulfur(VI) Fluoride Reactive Fragments
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00034 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 21, 2023 Category: Chemistry Authors: Arron Aatkar, Aini Vuorinen, Oliver E. Longfield, Katharine Gilbert, Rachel Peltier-Heap, Craig D. Wagner, Francesca Zappacosta, Katrin Rittinger, Chun-wa Chung, David House, Nicholas C. O. Tomkinson, and Jacob T. Bush Source Type: research

[ASAP] New High-Throughput Screen Discovers Novel Ligands of Full-Length Nuclear Receptor LRH ‑1
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00805 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 19, 2023 Category: Chemistry Authors: M. Merced Malabanan, Pratima Chapagain, Zeinab Haratipour, Woong Jae Choi, Abigail R. Orun, and Raymond D. Blind Source Type: research

[ASAP] Biosynthesis-Guided Discovery and Engineering of α‑Pyrone Natural Products from Type I Polyketide Synthases
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00081 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 19, 2023 Category: Chemistry Authors: Dongqi Yi and Vinayak Agarwal Source Type: research

[ASAP] Hematoxylin Nuclear Stain Reports Oxidative Stress via Near-Infrared Emission
ACS Chemical BiologyDOI: 10.1021/acschembio.3c00156 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 18, 2023 Category: Chemistry Authors: Rachel E. Langenbacher, Christopher P. Horoszko, Mijin Kim, and Daniel A. Heller Source Type: research

[ASAP] Biosynthesis of Antifungal Solanimycin May Involve an Iterative Nonribosomal Peptide Synthetase Module
ACS Chemical BiologyDOI: 10.1021/acschembio.2c00947 (Source: ACS Chemical Biology)
Source: ACS Chemical Biology - April 17, 2023 Category: Chemistry Authors: Annabel C. Murphy, Matthew Corney, Rita E. Monson, Miguel A. Matilla, George P. C. Salmond, and Finian J. Leeper Source Type: research