[ASAP] Discovery of a Novel Potent and Selective Calcium Release-Activated Calcium Channel Inhibitor: 2,6-Difluoro- < italic toggle="yes" > N < /italic > -(2 ′-methyl-3′-(4-methyl-5-oxo-4,5-dihydro-1,3,4-oxadiazol-2-yl)-[1,1′-biphenyl]-4-yl)benzamide. Structure–Activity Relationship and Preclinical Characterization
Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.1c01403
Source: Journal of Medicinal Chemistry - Category: Chemistry Authors: Nilesh Raghunath Khedkar, Nageswara Rao Irlapatti, Disha Dadke, Vijay Kanoje, Zubair Shaikh, Vijay Karche, Vikas Shinde, Gokul Deshmukh, Amit Patil, Santosh Jachak, Samiron Phukan, Praveenkumar Anidil Kizhakinagath, Milind Gholve, Trupti Bhankhede, Jagade Source Type: research