[ASAP] Highly Selective Sub-Nanomolar Cathepsin S Inhibitors by Merging Fragment Binders with Nitrile Inhibitors

Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.0c00949

Source: Journal of Medicinal Chemistry - September 17, 2020 Category: Chemistry Authors: Markus Schade, Beatrix Merla, Bernhard Lesch, Markus Wagener, Simone Timmermanns, Katrien Pletinckx, and Torsten Hertrampf Source Type: research