[ASAP] Covalent-Fragment Screening of BRD4 Identifies a Ligandable Site Orthogonal to the Acetyl-Lysine Binding Sites

ACS Chemical BiologyDOI: 10.1021/acschembio.0c00058

Source: ACS Chemical Biology - March 23, 2020 Category: Chemistry Authors: Michael D. Olp †, Daniel J. Sprague†, Christopher J. Goetz†, Stefan G. Kathman‡, Sarah L. Wynia-Smith†, Shifali Shishodia†, Steven B. Summers†, Ziyang Xu‡, Alexander V. Statsyuk‡¶, and Brian C. Smith*† Source Type: research