Optimization of Potent and Selective Tricyclic Indole Diazepinone Myeloid Cell Leukemia-1 Inhibitors Using Structure-Based Design

Journal of Medicinal ChemistryDOI: 10.1021/acs.jmedchem.7b01155

Source: Journal of Medicinal Chemistry - March 9, 2018 Category: Chemistry Authors: Subrata Shaw, Zhiguo Bian, Bin Zhao, James C. Tarr, Nagarathanam Veerasamy, Kyu Ok Jeon, Johannes Belmar, Allison L. Arnold, Stuart A. Fogarty, Evan Perry, John L. Sensintaffar, DeMarco V. Camper, Olivia W. Rossanese, Taekyu Lee, Edward T. Olejniczak and Source Type: research