Modification of the Orthosteric PPAR γ Covalent Antagonist Scaffold Yields an Improved Dual-Site Allosteric Inhibitor

ACS Chemical BiologyDOI: 10.1021/acschembio.6b01015

Source: ACS Chemical Biology - February 16, 2017 Category: Chemistry Authors: Richard Brust, Hua Lin, Jakob Fuhrmann, Alice Asteian, Theodore M. Kamenecka and Douglas J. Kojetin Source Type: research